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  1. 2025

  2. Synthesis of Secondary Amines of Bornylamine and Isobornylamine Containing a Saturated N-Heterocycle and Study of Their Antiviral Activity against Respiratory Syncytial Virus

    Tishchenko, S. A., Sokolova, A. S., Yarovaya, O. I., Krasnov, V. I., Shtro, A. A., Galochkina, A. V., Klabukov, A. M., Razgulyaeva, D. N. & Salakhutdinov, N. F., 27 Feb 2025, In: Russian Journal of General Chemistry. 95, 1, p. 79-87 9 p.

    Research output: Contribution to journal › Article › peer-review

  3. 2024

  4. Sulfide, Sulfoxide, and Sulfone Derivatives of Usnic Acid as Inhibitors of Human TDP1 and TDP2 Enzymes

    Filimonov, A. S., Mikhailova, M. A., Dyrkheeva, N. S., Chernyshova, I. A., Kornienko, T. E., Naumenko, K. A., Anarbaev, R. O., Nefedov, A. A., Achara, C., Curtis, A. D. M., Luzina, O. A., Volcho, K. P., Salakhutdinov, N. F., Lavrik, O. I. & Reynisson, J., 17 Dec 2024, In: Chemistry (Switzerland). 6, 6, p. 1658-1679 22 p.

    Research output: Contribution to journal › Article › peer-review

  5. Antidiabetic Effect of Dihydrobetulonic Acid Derivatives as Pparα/γ Agonists

    Khvostov, M. V., Blokhin, M. E., Borisov, S. A., Fomenko, V. V., Meshkova, Y. V., Zhukova, N. A., Nikonova, S. V., Pavlova, S. V., Pogosova, M. A., Medvedev, S. P., Luzina, O. A. & Salakhutdinov, N. F., 5 Dec 2024, In: Scientia Pharmaceutica. 92, 4, 65.

    Research output: Contribution to journal › Article › peer-review

  6. Novel Peptide–Drug Conjugates with Dual Anticancer Activity

    O’Flaherty, S., Luzina, O. A., Dyrkheeva, N. S., Krier, Y., Leprince, J., Zakharenko, A. L., Pokrovsky, M. A., Pokrovsky, A. G., Lavrik, O. I., Salakhutdinov, N. F., Varbanov, M., Devocelle, M. & Volcho, K. P., 19 Nov 2024, In: International Journal of Molecular Sciences. 25, 22, 12411.

    Research output: Contribution to journal › Article › peer-review

  7. (+)-fenchol and (−)-isopinocampheol derivatives targeting the entry process of filoviruses

    Sokolova, A. S., Baev, D. S., Mordvinova, E. D., Yarovaya, O. I., Volkova, N. V., Shcherbakov, D. N., Okhina, A. A., Rogachev, A. D., Shnaider, T. A., Chvileva, A. S., Nikitina, T. V., Tolstikova, T. G. & Salakhutdinov, N. F., 5 Sept 2024, In: European Journal of Medicinal Chemistry. 275, 16 p., 116596.

    Research output: Contribution to journal › Article › peer-review

  8. Pharmacokinetics and Dose Proportionality Study of a Novel Antiparkinsonian Agent, a 1H-1,2,4-Triazol-3-ylthio-conjugate of Prottremine

    Gorina, D. S., Lastovka, A. V., Rogachev, A. D., Podturkina, A. V., Pavlova, A. V., Ardashov, O. V., Li-Zhulanov, N. S., Tolstikova, T. G., Volcho, K. P. & Salakhutdinov, N. F., Sept 2024, In: Molecules. 29, 18, 4498.

    Research output: Contribution to journal › Article › peer-review

  9. The first non-symmetrically substituted conjugates of bispidine with monoterpenoids and amino acids. Synthesis and application for catalysis of addition of diethylzinc to aldehydes

    Ponomarev, K. Y., Mozhaitsev, E. S., Li-Zhulanov, N. S., Okhina, A. A., Nefedov, A. A., Rogachev, A. D., Suslov, E. V., Dalinger, A. I., Vatsadze, S. Z., Volcho, K. P. & Salakhutdinov, N. F., Aug 2024, In: Russian Chemical Bulletin. 73, 8, p. 2248-2260 13 p.

    Research output: Contribution to journal › Article › peer-review

  10. 2-Aryl-1-hydroxyimidazoles possessing antiviral activity against a wide range of orthopoxviruses, including the variola virus

    Басанова, Е. И., Куликова, Е. А., Бормотов, Н. И., Серова, О. А., Шишкина, Л. Н., Овчинникова, А. С., Одношевский, Д. А., Пьянков, О. В., Агафонов, А. П., Яровая, О. И., Борисевич, С. С., Ильина, М. Г., Колыбалов, Д. С., Архипов, С. Г., Богданов, Н. Е., Павлова, М. А., Салахутдинов, Н. Ф., Перевалов, В. П. & Никитина, П. А., 5 Jul 2024, In: RSC Medicinal Chemistry. 15, 9, p. 3196-3211 16 p.

    Research output: Contribution to journal › Article › peer-review

  11. Производные имидазолидин-2,4-диона и имидазолидин-2,4,5-триона на основе смоляных кислот, проявляющие антиинвазивную активность в отношении клеток глиобластомы линий T98G и SNB19

    Чересиз, С. В., Ковалева, К. С., Яровая, О. И., Салахутдинов, Н. Ф. & Покровский, А. Г., 17 Jun 2024, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2821104, 8 Dec 2023, Priority date 8 Dec 2023, Priority No. 2023132332

    Research output: Patent › Patent for invention

  12. Global LC-MS/MS targeted metabolomics using a combination of HILIC and RP LC separation modes on an organic monolithic column based on 1-vinyl-1,2,4-triazole

    Basov, N. V., Rogachev, A. D., Aleshkova, M. A., Gaisler, E. V., Sotnikova, Y. S., Patrushev, Y. V., Tolstikova, T. G., Yarovaya, O. I., Pokrovsky, A. G. & Salakhutdinov, N. F., 15 Jan 2024, In: Talanta. 267, 125168.

    Research output: Contribution to journal › Article › peer-review

  13. 2023

  14. A Novel 3-meta-Pyridine-1,2,4-oxadiazole Derivative of Glycyrrhetinic Acid as a Safe and Promising Candidate for Overcoming P-Glycoprotein-Mediated Multidrug Resistance in Tumor Cells

    Moralev, A. D., Salomatina, O. V., Chernikov, I. V., Salakhutdinov, N. F., Zenkova, M. A. & Markov, A. V., 26 Dec 2023, In: ACS Omega. 8, 51, p. 48813-48824 12 p.

    Research output: Contribution to journal › Article › peer-review

  15. Synthesis of Norabietyl and Nordehydroabietyl Imidazolidine-2,4,5-Triones and Their Activity against Tyrosyl-DNA Phosphodiesterase 1

    Kovaleva, K. S., Yarovaya, O. I., Chernyshova, I. A., Zakharenko, A. L., Cheresiz, S. V., Azimirad, A., Pokrovsky, A. G., Lavrik, O. I. & Salakhutdinov, N. F., Dec 2023, In: MolBank. 2023, 4, М1743.

    Research output: Contribution to journal › Article › peer-review

  16. Pharmacokinetic study of Tdp1 inhibitor resulted in a significant increase in antitumor effect in the treatment of Lewis lung carcinoma in mice by its combination with topotecan

    Okhina, A. A., Kornienko, T. E., Rogachev, A. D., Luzina, O. A., Popova, N. A., Nikolin, V. P., Zakharenko, A. L., Dyrkheeva, N. S., Pokrovsky, A. G., Salakhutdinov, N. F. & Lavrik, O. I., 30 Nov 2023, In: Journal of Pharmaceutical and Biomedical Analysis. 236, 9 p., 115731.

    Research output: Contribution to journal › Article › peer-review

  17. Chiral N-(dialkyloctahydro-2H-chromen-4-yl)acetamides: synthesis and analgesic activity

    Li-Zhulanov, N. S., Kuznetsova, V. A., Gatilov, Y. V., Volcho, K. P., Khvostov, M. V., Tolstikova, T. G. & Salakhutdinov, N. F., Oct 2023, In: Russian Chemical Bulletin. 72, 10, p. 2430-2438 9 p.

    Research output: Contribution to journal › Article › peer-review

  18. Development of an LC-MS/MS-based method for quantification and pharmacokinetics study on SCID mice of a dehydroabietylamine-adamantylamine conjugate, a promising inhibitor of the DNA repair enzyme

    Okhina, A. A., Rogachev, A. D., Kovaleva, K. S., Yarovaya, O. I., Khotskina, A. S., Zavyalov, E. L., Vatsadze, S. Z., Pokrovsky, A. G. & Salakhutdinov, N. F., 20 Sept 2023, In: Journal of Pharmaceutical and Biomedical Analysis. 234, 115507.

    Research output: Contribution to journal › Article › peer-review

  19. Chiral N-(Octahydro-2H-chromen-4-yl)-2-(dialkylamino)acetamides: Synthesis and Analgesic Activity

    Li-Zhulanov, N. S., Nikolaichuk, K. M., Gatilov, Y. V., Volcho, K. P., Khvostov, M. V., Tolstikova, T. G. & Salakhutdinov, N. F., Sept 2023, In: Doklady Chemistry. 512, 1, p. 242-248 7 p.

    Research output: Contribution to journal › Article › peer-review

  20. Effect of Usnic Acid-Derived Tyrosyl-DNA Phosphodiesterase 1 Inhibitor Used as Monotherapy or in Combination with Olaparib on Transplanted Tumors In Vivo

    Kornienko, T. E., Zakharenko, A. L., Ilina, E. S., Chepanova, A. A., Zakharova, O. D., Dyrkheeva, N. S., Popova, N. A., Nikolin, V. P., Filimonov, A. S., Luzina, O. A., Salakhutdinov, N. F. & Lavrik, O. I., Apr 2023, In: Molecular Biology. 57, 2, p. 214-224 11 p.

    Research output: Contribution to journal › Article › peer-review

  21. Transcriptomic Analysis of CRISPR/Cas9-Mediated PARP1-Knockout Cells under the Influence of Topotecan and TDP1 Inhibitor

    Dyrkheeva, N. S., Malakhova, A. A., Zakharenko, A. L., Okorokova, L. S., Shtokalo, D. N., Pavlova, S. V., Medvedev, S. P., Zakian, S. M., Nushtaeva, A. A., Tupikin, A. E., Kabilov, M. R., Khodyreva, S. N., Luzina, O. A., Salakhutdinov, N. F. & Lavrik, O. I., 7 Mar 2023, In: International Journal of Molecular Sciences. 24, 6, 5148.

    Research output: Contribution to journal › Article › peer-review

  22. Влияние производного усниновой кислоты (ингибитора тирозил-ДНК-фосфодиэстеразы 1) на трансплантированные опухоли in vivo в качестве монотерапии и в сочетании с олапарибом

    Kornienko, T. E., Zakharenko, A. L., Ilina, E. S., Chepanova, A. A., Zakharova, O. D., Dyrkheeva, N. S., Popova, N. A., Nikolin, V. P., Filimonov, A. S., Luzina, O. A., Salakhutdinov, N. F. & Lavrik, O. I., 1 Mar 2023, In: Molekuliarnaia biologiia. 57, 2, p. 220-231 12 p., 8.

    Research output: Contribution to journal › Article › peer-review

  23. Synthesis of a Novel 9-O Berberine Derivative and Evaluation of Its Hypoglycemic Effect

    Gladkova, E. D., Valutsa, N., Borisov, S. A., Khvostov, M. V., Luzina, O. A., Tolstikova, T. G. & Salakhutdinov, N. F., Mar 2023, In: MolBank. 2023, 1, М1597.

    Research output: Contribution to journal › Article › peer-review

  24. Synthesis of N-heterocyclic amides based on (+)-camphoric acid and study of their antiviral activity and pharmacokinetics

    Yarovaya, O. I., Baranova, D. V., Sokolova, A. S., Nemolochnova, A. G., Sal'nikova, O. P., Fat'anova, A. V., Rogachev, A. D., Volobueva, A. S., Zarubaev, V. V., Pokrovsky, A. G. & Salakhutdinov, N. F., Mar 2023, In: Russian Chemical Bulletin. 72, 3, p. 807-818 12 p.

    Research output: Contribution to journal › Article › peer-review

  25. Novel TDP1 Inhibitors: Disubstituted Thiazolidine-2,4-Diones Containing Monoterpene Moieties

    Ivankin, D. I., Kornienko, T. E., Mikhailova, M. A., Dyrkheeva, N. S., Zakharenko, A. L., Achara, C., Reynisson, J., Golyshev, V. M., Luzina, O. A., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 14 Feb 2023, In: International Journal of Molecular Sciences. 24, 4, 3834.

    Research output: Contribution to journal › Article › peer-review

  26. 9-N-n-alkyl Berberine Derivatives: Hypoglycemic Activity Evaluation

    Khvostov, M. V., Gladkova, E. D., Borisov, S. A., Fedotova, M. S., Zhukova, N. A., Marenina, M. K., Meshkova, Y. V., Valutsa, N., Luzina, O. A., Tolstikova, T. G. & Salakhutdinov, N. F., 1 Jan 2023, In: Pharmaceutics. 15, 1, 44.

    Research output: Contribution to journal › Article › peer-review

  27. Structure-Based Design, Synthesis, and Biological Evaluation of the Cage-Amide Derived Orthopox Virus Replication Inhibitors

    Mozhaitsev, E. S., Suslov, E. V., Rastrepaeva, D. A., Yarovaya, O. I., Borisevich, S. S., Khamitov, E. M., Kolybalov, D. S., Arkhipov, S. G., Bormotov, N. I., Shishkina, L. N., Serova, O. A., Brunilin, R. V., Vernigora, A. A., Nawrozkij, M. B., Agafonov, A. P., Maksyutov, R. A., Volcho, K. P. & Salakhutdinov, N. F., 1 Jan 2023, In: Viruses. 15, 1, 29.

    Research output: Contribution to journal › Article › peer-review

  28. Synthesis of conjugates of (aR,7S)-colchicine with monoterpenoids and investigation of their biological activity

    Shchegravina, E. S., Usova, S. D., Baev, D. S., Mozhaitsev, E. S., Shcherbakov, D. N., Belenkaya, S. V., Volosnikova, E. A., Chirkova, V. Y., Sharlaeva, E. A., Svirshchevskaya, E. V., Fonareva, I. P., Sitdikova, A. R., Salakhutdinov, N. F., Yarovaya, O. I. & Fedorov, A. Y., 1 Jan 2023, In: Russian Chemical Bulletin. 72, 1, p. 248-262 15 p.

    Research output: Contribution to journal › Article › peer-review

  29. Synthesis of non-symmetric N-benzylbispidinol amides and study of their inhibitory activity against the main protease of the SARS-CoV-2 virus

    Dalinger, A. I., Baev, D. S., Yarovaya, O. I., Chirkova, V. Y., Sharlaeva, E. A., Belenkaya, S. V., Shcherbakov, D. N., Salakhutdinov, N. F. & Vatsadze, S. Z., 1 Jan 2023, In: Russian Chemical Bulletin. 72, 1, p. 239-247 9 p.

    Research output: Contribution to journal › Article › peer-review

  30. Corrigendum: The main protease 3CLpro of the SARS-CoV-2 virus: how to turn an enemy into a helper

    Belenkaya, S. V., Merkuleva, I. A., Yarovaya, O. I., Chirkova, V. Y., Sharlaeva, E. A., Shanshin, D. V., Volosnikova, E. A., Vatsadze, S. Z., Khvostov, M. V., Salakhutdinov, N. F. & Shcherbakov, D., 2023, In: Frontiers in Bioengineering and Biotechnology. 11, 1294266.

    Research output: Contribution to journal › Article › peer-review

  31. The main protease 3CLpro of the SARS-CoV-2 virus: how to turn an enemy into a helper

    Belenkaya, S. V., Merkuleva, I. A., Yarovaya, O. I., Chirkova, V. Y., Sharlaeva, E. A., Shanshin, D. V., Volosnikova, E. A., Vatsadze, S. Z., Khvostov, M. V., Salakhutdinov, N. F. & Shcherbakov, D. N., 2023, In: Frontiers in Bioengineering and Biotechnology. 11, 1187761.

    Research output: Contribution to journal › Article › peer-review

  32. 2022

  33. (1S,5R)-6,6-Dimethyl-4-(((1S,2S,5S)-2,6,6-trimethyl-4-oxobicyclo[3.1.1]heptan-2-yl)methyl)bicyclo[3.1.1]hept-3-en-2-one

    Ardashov, O. V., Korchagina, D. V., Bagryanskaya, I. Y., Volcho, K. P. & Salakhutdinov, N. F., 1 Dec 2022, In: MolBank. 2022, 4, M1465.

    Research output: Contribution to journal › Article › peer-review

  34. A Newly Identified Monoterpenoid-Based Small Molecule Able to Support the Survival of Primary Cultured Dopamine Neurons and Alleviate MPTP-Induced Toxicity In Vivo

    Kotliarova, A., Podturkina, A. V., Pavlova, A. V., Gorina, D. S., Lastovka, A. V., Ardashov, O. V., Rogachev, A. D., Izyurov, A. E., Arefieva, A. B., Kulikov, A. V., Tolstikova, T. G., Volcho, K. P., Salakhutdinov, N. F. & Sidorova, Y., Dec 2022, In: Molecules. 27, 23, 8286.

    Research output: Contribution to journal › Article › peer-review

  35. Study of Hypoglycemic Activity of Novel 9-N-alkyltetrahydroberberine Derivatives

    Khvostov, M. V., Gladkova, E. D., Borisov, S. A., Fedotova, M. S., Zhukova, N. A., Marenina, M. K., Meshkova, Y. V., Luzina, O. A., Tolstikova, T. G. & Salakhutdinov, N. F., Nov 2022, In: International Journal of Molecular Sciences. 23, 22, 14186.

    Research output: Contribution to journal › Article › peer-review

  36. Nitrogen-Containing Heterocyclic Compounds Obtained from Monoterpenes or Their Derivatives: Synthesis and Properties

    Chernyshov, V. V., Popadyuk, I. I., Yarovaya, O. I. & Salakhutdinov, N. F., Oct 2022, In: Topics in current chemistry (Cham). 380, 5, p. 42 1 p., 42.

    Research output: Contribution to journal › Review article › peer-review

  37. Stability Study, Quantification Method and Pharmacokinetics Investigation of a Coumarin-Monoterpene Conjugate Possessing Antiviral Properties against Respiratory Syncytial Virus

    Nemolochnova, A. G., Rogachev, A. D., Salnikova, O. P., Khomenko, T. M., Volcho, K. P., Yarovaya, O. I., Fatianova, A. V., Pokrovsky, A. G. & Salakhutdinov, N. F., 18 Sept 2022, In: Pharmaceuticals. 15, 9, 1158.

    Research output: Contribution to journal › Article › peer-review

  38. Determination of elemental impurities Cd, Pb, As, Hg, Co, V, Ni, Pd, Ru, Ag, Pt, Mo, Al, and Fe in highly potent analgesic activity agent by microwave-induced plasma optical emission spectrometry (MIP OES)

    Zubricheva, D. V., Lastovka, A. V., Il’ina, I. V., Volcho, K. P., Tikhova, V. D., Fadeeva, V. P. & Salakhutdinov, N. F., Sept 2022, In: Chemical Papers. 76, 9, p. 5677-5689 13 p.

    Research output: Contribution to journal › Article › peer-review

  39. Synthesis and Antiviral Properties of Camphor-Derived Iminothiazolidine-4-Ones and 2,3-Dihydrothiazoles

    Oreshko, V. V., Kovaleva, K. S., Mordvinova, E. D., Yarovaya, O. I., Gatilov, Y. V., Shcherbakov, D. N., Bormotov, N. I., Serova, O. A., Shishkina, L. N. & Salakhutdinov, N. F., Aug 2022, In: Molecules. 27, 15, 4761.

    Research output: Contribution to journal › Article › peer-review

  40. Design, Synthesis, and Biological Evaluation of (+)-Camphor- and (−)-Fenchone-Based Derivatives as Potent Orthopoxvirus Inhibitors

    Sokolova, A. S., Kovaleva, K. S., Kuranov, S. O., Bormotov, N. I., Borisevich, S. S., Zhukovets, A. A., Yarovaya, O. I., Serova, O. A., Nawrozkij, M. B., Vernigora, A. A., Davidenko, A. V., Khamitov, E. M., Peshkov, R. Y., Shishkina, L. N., Maksuytov, R. A. & Salakhutdinov, N. F., 20 Jun 2022, In: ChemMedChem. 17, 12, p. e202100771 26 p., e202100771.

    Research output: Contribution to journal › Article › peer-review

  41. Novel Epoxides of Soloxolone Methyl: An Effect of the Formation of Oxirane Ring and Stereoisomerism on Cytotoxic Profile, Anti-Metastatic and Anti-Inflammatory Activities In Vitro and In Vivo

    Salomatina, O. V., Sen’kova, A. V., Moralev, A. D., Savin, I. A., Komarova, N. I., Salakhutdinov, N. F., Zenkova, M. A. & Markov, A. V., 1 Jun 2022, In: International Journal of Molecular Sciences. 23, 11, 6214.

    Research output: Contribution to journal › Article › peer-review

  42. Novel Soloxolone Amides as Potent Anti-Glioblastoma Candidates: Design, Synthesis, In Silico Analysis and Biological Activities In Vitro and In Vivo

    Markov, A. V., Ilyina, A. A., Salomatina, O. V., Sen’kova, A. V., Okhina, A. A., Rogachev, A. D., Salakhutdinov, N. F. & Zenkova, M. A., May 2022, In: Pharmaceuticals. 15, 5, 603.

    Research output: Contribution to journal › Article › peer-review

  43. Inhibition of the DNA repair enzyme TDP1 by the resin acid derivatives as a new way to increase the efficiency of glioblastoma chemotherapy

    Kovaleva, K., Oleshko, O., Yarovaya, O., Cheresiz, S., Zakharenko, A., Ponomarev, K., Lavrik, O., Pokrovsky, A. & Salakhutdinov, N., 4 Feb 2022, Actual Problems of Organic Chemistry and Biotechnology, OCBT 2020: Proceedings of the International Scientific Conference. Bakulev, V., Kovaleva, E., Glukhareva, T., Beryozkina, T., Schafran, Y., Lyubyakina, P. & Koptyaeva, O. (eds.). American Institute of Physics Inc., 020036. (AIP Conference Proceedings; vol. 2390).

    Research output: Chapter in Book/Report/Conference proceeding › Conference contribution › Research › peer-review

  44. MPTP-Treated Zebrafish Recapitulate ‘Late-Stage’ Parkinson’s-like Cognitive Decline

    Bashirzade, A. A. O., Cheresiz, S. V., Belova, A. S., Drobkov, A. V., Korotaeva, A. D., Azizi-Arani, S., Azimirad, A., Odle, E., Gild, E. Y. V., Ardashov, O. V., Volcho, K. P., Bozhko, D. V., Myrov, V. O., Kolchanova, S. M., Polovian, A. I., Galumov, G. K., Salakhutdinov, N. F., Amstislavskaya, T. G. & Kalueff, A. V., Feb 2022, In: Toxics. 10, 2, 69.

    Research output: Contribution to journal › Article › peer-review

  45. Design and Evaluation of Bispidine-Based SARS-CoV-2 Main Protease Inhibitors

    Shcherbakov, D., Baev, D., Kalinin, M., Dalinger, A., Chirkova, V., Belenkaya, S., Khvostov, A., Krut'Ko, D., Medved'Ko, A., Volosnikova, E., Sharlaeva, E., Shanshin, D., Tolstikova, T., Yarovaya, O., Maksyutov, R., Salakhutdinov, N. & Vatsadze, S., 13 Jan 2022, In: ACS Medicinal Chemistry Letters. 13, 1, p. 140-147 8 p.

    Research output: Contribution to journal › Article › peer-review

  46. Synthesis and In Vitro Study of Antiviral Activity of Glycyrrhizin Nicotinate Derivatives against HIV-1 Pseudoviruses and SARS-CoV-2 Viruses

    Fomenko, V. V., Rudometova, N. B., Yarovaya, O. I., Rogachev, A. D., Fando, A. A., Zaykovskaya, A. V., Komarova, N. I., Shcherbakov, D. N., Pyankov, O. V., Pokrovsky, A. G., Karpenko, L. I., Maksyutov, R. A. & Salakhutdinov, N. F., 1 Jan 2022, In: Molecules. 27, 1, 295.

    Research output: Contribution to journal › Article › peer-review

  47. 2021

  48. Novel bispidine-monoterpene conjugates—Synthesis and application as ligands for the catalytic ethylation of chalcones

    Suslov, E. V., Ponomarev, K. Y., Patrusheva, O. S., Kuranov, S. O., Okhina, A. A., Rogachev, A. D., Munkuev, A. A., Ottenbacher, R. V., Dalinger, A. I., Kalinin, M. A., Vatsadze, S. Z., Volcho, K. P. & Salakhutdinov, N. F., 1 Dec 2021, In: Molecules. 26, 24, 7539.

    Research output: Contribution to journal › Article › peer-review

  49. Stereoselective Cycloaddition of Alkanesulfonyl Chlorides to Dihydroberberine

    Gladkova, E. D., Luzina, O. A. & Salakhutdinov, N. F., 18 Nov 2021, In: Chemistry of Natural Compounds. 57, 6, p. 1062-1065 4 p.

    Research output: Contribution to journal › Article › peer-review

  50. New hybrid compounds combining fragments of usnic acid and thioether are inhibitors of human enzymes TDP1, TDP2 and PARP1

    Dyrkheeva, N. S., Filimonov, A. S., Luzina, O. A., Orlova, K. A., Chernyshova, I. A., Kornienko, T. E., Malakhova, A. A., Medvedev, S. P., Zakharenko, A. L., Ilina, E. S., Anarbaev, R. O., Naumenko, K. N., Klabenkova, K. V., Burakova, E. A., Stetsenko, D. A., Zakian, S. M., Salakhutdinov, N. F. & Lavrik, O. I., 1 Nov 2021, In: International Journal of Molecular Sciences. 22, 21, 11336.

    Research output: Contribution to journal › Article › peer-review

  51. Dehydroabietylamine-based thiazolidin-4-ones and 2-thioxoimidazolidin-4-ones as novel tyrosyl-DNA phosphodiesterase 1 inhibitors

    Kovaleva, K., Mamontova, E., Yarovaya, O., Zakharova, O., Zakharenko, A., Lavrik, O. & Salakhutdinov, N., Nov 2021, In: Molecular Diversity. 25, 4, p. 2389-2397 9 p.

    Research output: Contribution to journal › Article › peer-review

  52. Stability study of the antiviral agent camphecene in dried blood spots at different temperatures

    Okhina, A. A., Rogachev, A. D., Yarovaya, O. I., Pokrovsky, A. G. & Salakhutdinov, N. F., Oct 2021, In: Drug Testing and Analysis. 13, 10, p. 1797-1802 6 p.

    Research output: Contribution to journal › Letter › peer-review

  53. The influence of an enamine usnic acid derivative (a tyrosyl-DNA phosphodiesterase 1 inhibitor) on the therapeutic effect of topotecan against transplanted tumors in vivo

    Nikolin, V. P., Popova, N. A., Kaledin, V. I., Luzina, O. A., Zakharenko, A. L., Salakhutdinov, N. F. & Lavrik, O. I., Oct 2021, In: Clinical and Experimental Metastasis. 38, 5, p. 431-440 10 p.

    Research output: Contribution to journal › Article › peer-review

  54. New hybrid compounds combining fragments of usnic acid and monoterpenoids for effective tyrosyl-dna phosphodiesterase 1 inhibition

    Dyrkheeva, N. S., Filimonov, A. S., Luzina, O. A., Zakharenko, A. L., Ilina, E. S., Malakhova, A. A., Medvedev, S. P., Reynisson, J., Volcho, K. P., Zakian, S. M., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jul 2021, In: Biomolecules. 11, 7, 973.

    Research output: Contribution to journal › Article › peer-review

  55. Biostability study, quantitation method and preliminary pharmacokinetics of a new antifilovirus agent based on borneol and 3-(piperidin-1-yl)propanoic acid

    Rogachev, A. D., Putilova, V. P., Zaykovskaya, A. V., Yarovaya, O. I., Sokolova, A. S., Fomenko, V. V., Pyankov, O. V., Maksyutov, R. A., Pokrovsky, A. G. & Salakhutdinov, N. F., 30 May 2021, In: Journal of Pharmaceutical and Biomedical Analysis. 199, 114062.

    Research output: Contribution to journal › Article › peer-review

  56. New class of hantaan virus inhibitors based on conjugation of the isoindole fragment to (+)-camphor or (−)-fenchone hydrazonesv

    Yarovaya, O. I., Kovaleva, K. S., Zaykovskaya, A. A., Yashina, L. N., Scherbakova, N. S., Scherbakov, D. N., Borisevich, S. S., Zubkov, F. I., Antonova, A. S., Peshkov, R. Y., Eltsov, I. V., Pyankov, O. V., Maksyutov, R. A. & Salakhutdinov, N. F., 15 May 2021, In: Bioorganic and Medicinal Chemistry Letters. 40, 127926.

    Research output: Contribution to journal › Article › peer-review

  57. Design, synthesis, and molecular docking study of new tyrosyl-dna phosphodiesterase 1 (Tdp1) inhibitors combining resin acids and adamantane moieties

    Kovaleva, K., Yarovaya, O., Ponomarev, K., Cheresiz, S., Azimirad, A., Chernyshova, I., Zakharenko, A., Konev, V., Khlebnikova, T., Mozhaytsev, E., Suslov, E., Nilov, D., Švedas, V., Pokrovsky, A., Lavrik, O. & Salakhutdinov, N., 1 May 2021, In: Pharmaceuticals. 14, 5, 422.

    Research output: Contribution to journal › Article › peer-review

  58. Discovery of Novel Sultone Fused Berberine Derivatives as Promising Tdp1 Inhibitors

    Gladkova, E. D., Chepanova, A. A., Ilina, E. S., Zakharenko, A. L., Reynisson, J., Luzina, O. A., Volcho, K. P., Lavrik, O. I. & Salakhutdinov, N. F., 30 Mar 2021, In: Molecules (Basel, Switzerland). 26, 7, 1945.

    Research output: Contribution to journal › Article › peer-review

  59. Противоопухлевая активность комбинации топотекана и ингибитора тирозил-ДНК-фосфодиэстеразы 1 на модели асцитной карциномы Кребс-2 мыши

    Dyrkheeva, N. S., Zakharenko, A. L., Novoselova, E. S., Chepanova, A. A., Popova, N. A., Nikolin, V. P., Luzina, O. A., Salakhutdinov, N. F., Ryabchikova, E. I. & Lavrik, O. I., 1 Mar 2021, In: Molekuliarnaia biologiia. 55, 2, p. 312-317 6 p., 12.

    Research output: Contribution to journal › Article › peer-review

  60. Antitumor Activity of the Combination of Topotecan and Tyrosyl-DNA-Phosphodiesterase 1 Inhibitor on Model Krebs-2 Mouse Ascite Carcinoma

    Dyrkheeva, N. S., Zakharenko, A. L., Novoselova, E. S., Chepanova, A. A., Popova, N. A., Nikolin, V. P., Luzina, O. A., Salakhutdinov, N. F., Ryabchikova, E. I. & Lavrik, O. I., Mar 2021, In: Molecular Biology. 55, 2, p. 273-277 5 p.

    Research output: Contribution to journal › Article › peer-review

  61. Unexpected Ring Opening During the Imination of Camphor-Type Bicyclic Ketones

    Chernyshov, V. V., Yarovaya, O. I., Vatsadze, S. Z., Borisevich, S. S., Trukhan, S. N., Gatilov, Y. V., Peshkov, R. Y., Eltsov, I. V., Martyanov, O. N. & Salakhutdinov, N. F., 22 Jan 2021, In: European Journal of Organic Chemistry. 2021, 3, p. 452-463 12 p.

    Research output: Contribution to journal › Article › peer-review

  62. 2020

  63. Monoterpenoid-based inhibitors of filoviruses targeting the glycoprotein-mediated entry process

    Sokolova, A. S., Yarovaya, O. I., Zybkina, A. V., Mordvinova, E. D., Shcherbakova, N. S., Zaykovskaya, A. V., Baev, D. S., Tolstikova, T. G., Shcherbakov, D. N., Pyankov, O. V., Maksyutov, R. A. & Salakhutdinov, N. F., 1 Dec 2020, In: European Journal of Medicinal Chemistry. 207, 17 p., 112726.

    Research output: Contribution to journal › Article › peer-review

  64. The first berberine-based inhibitors of tyrosyl-dna phosphodiesterase 1 (Tdp1), an important dna repair enzyme

    Gladkova, E. D., Nechepurenko, I. V., Bredikhin, R. A., Chepanova, A. A., Zakharenko, A. L., Luzina, O. A., Ilina, E. S., Dyrkheeva, N. S., Mamontova, E. M., Anarbaev, R. O., Reynisson, J., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Oct 2020, In: International Journal of Molecular Sciences. 21, 19, p. 1-16 16 p., 7162.

    Research output: Contribution to journal › Article › peer-review

  65. New chemical agents based on adamantane-monoterpene conjugates against orthopoxvirus infections

    Suslov, E. V., Mozhaytsev, E. S., Korchagina, D. V., Bormotov, N. I., Yarovaya, O. I., Volcho, K. P., Serova, O. A., Agafonov, A. P., Maksyutov, R. A., Shishkina, L. N. & Salakhutdinov, N. F., Oct 2020, In: RSC Medicinal Chemistry. 11, 10, p. 1185-1195 11 p.

    Research output: Contribution to journal › Article › peer-review

  66. Menthylamine synthesis via gold-catalyzed hydrogenation of menthone oxime

    Demidova, Y. S., Mozhaitsev, E. S., Suslov, E. V., Nefedov, A. A., Saraev, A. A., Volcho, K. P., Salakhutdinov, N. F., Simakov, A., Simakova, I. L. & Murzin, D. Y., 5 Sept 2020, In: Applied Catalysis A: General. 605, 10 p., 117799.

    Research output: Contribution to journal › Article › peer-review

  67. Usnic Acid Conjugates with Monoterpenoids as Potent Tyrosyl-DNA Phosphodiesterase 1 Inhibitors

    Luzina, O., Filimonov, A., Zakharenko, A., Chepanova, A., Zakharova, O., Ilina, E., Dyrkheeva, N., Likhatskaya, G., Salakhutdinov, N. & Lavrik, O., 28 Aug 2020, In: Journal of Natural Products. 83, 8, p. 2320-2329 10 p.

    Research output: Contribution to journal › Article › peer-review

  68. Design, Synthesis, and Biological Investigation of Novel Classes of 3-Carene-Derived Potent Inhibitors of TDP1

    Il'ina, I. V., Dyrkheeva, N. S., Zakharenko, A. L., Sidorenko, A. Y., Li-Zhulanov, N. S., Korchagina, D. V., Chand, R., Ayine-Tora, D. M., Chepanova, A. A., Zakharova, O. D., Ilina, E. S., Reynisson, J., Malakhova, A. A., Medvedev, S. P., Zakian, S. M., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., Aug 2020, In: Molecules (Basel, Switzerland). 25, 15, 22 p., 3496.

    Research output: Contribution to journal › Article › peer-review

  69. Synthesis of 1,3-Oxazine Derivatives Based on (–)-Isopulegol using the Ritter Reaction and Study of their Analgesic Activity

    Li-Zhulanov, N. S., Pavlova, A. V., Korchagina, D. V., Gatilov, Y. V., Volcho, K. P., Tolstikova, T. G. & Salakhutdinov, N. F., 1 Jul 2020, In: Chemistry of Heterocyclic Compounds. 56, 7, p. 936-941 6 p.

    Research output: Contribution to journal › Article › peer-review

  70. Synthesis of Fluorinated Octahydro-2H-Chromenes in the Presence of the BF3·Et2O–H2O Catalytic System

    Il’ina, I. V., Patrusheva, O. S., Korchagina, D. V., Volcho, K. P. & Salakhutdinov, N. F., 1 Jul 2020, In: Chemistry of Heterocyclic Compounds. 56, 7, p. 867-874 8 p.

    Research output: Contribution to journal › Article › peer-review

  71. Synthesis of isobenzofuran derivatives from renewable 2-carene over halloysite nanotubes

    Sidorenko, A. Y., Kravtsova, A. V., Mäki-Arvela, P., Aho, A., Sandberg, T., Il'ina, I. V., Li-Zhulanov, N. S., Korchagina, D. V., Volcho, K. P., Salakhutdinov, N. F., Murzin, D. Y. & Agabekov, V. E., Jul 2020, In: Molecular Catalysis. 490, 8 p., 110974.

    Research output: Contribution to journal › Article › peer-review

  72. 1,1’-(Гексан-1,6-диил)бис(3-(((1R,4aS,10aR)-7-изопропил-1,4a-диметил-1,2,3,4,4a,9,10,10a-октагидрофенантрен-1-ил)метил)мочевина, проявляющая ингибирующее действие в отношении фермента тирозил-ДНК-фосфодиэстеразы 1 человека и увеличивающая активность темозоломида в отношении клеток глиобластомы

    Ковалева, К. С., Олешко, О. С., Яровая, О. И., Мамонтова, Е. М., Захаренко, А. Л., Захарова, О. Д., Чересиз, С. В., Покровский, А. Г., Лаврик, О. И. & Салахутдинов, Н. Ф., 26 Jun 2020, IPC No. C07C275/24, A61K31/17, A61P35/00, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2724882, Priority date 28 Nov 2019, Priority No. 2019138671

    Research output: Patent › Patent for invention

  73. Synthesis of cyclic D-(+)-camphoric acid imides and study of their antiviral activity

    Chernyshov, V. V., Yarovaya, O. I., Peshkov, R. Y. & Salakhutdinov, N. F., 1 Jun 2020, In: Chemistry of Heterocyclic Compounds. 56, 6, p. 763-768 6 p.

    Research output: Contribution to journal › Article › peer-review

  74. Stereoselectivity Inversion by Water Addition in the −SO3H-catalyzed Tandem Prins-Ritter Reaction for Synthesis of 4-amidotetrahydropyran Derivatives

    Sidorenko, A. Y., Li-Zhulanov, N. S., Mäki-Arvela, P., Sandberg, T., Kravtsova, A. V., Peixoto, A. F., Freire, C., Volcho, K. P., Salakhutdinov, N. F., Agabekov, V. E. & Murzin, D. Y., 7 May 2020, In: ChemCatChem. 12, 9, p. 2605-2609 5 p.

    Research output: Contribution to journal › Article › peer-review

  75. Analytical Control of Impurities and Active Ingredients in a (–)-Isopulegol Derivative with Highly Potent Analgesic Activity

    Lastovka, A. V., Fedeeva, V. P., Il’ina, I. V. & Salakhutdinov, N. F., 1 May 2020, In: Pharmaceutical Chemistry Journal. 54, 2, p. 190-194 5 p.

    Research output: Contribution to journal › Article › peer-review

  76. Catalytic synthesis of bioactive 2H-chromene alcohols from (−)-isopulegol and acetone on sulfonated clays

    Laluc, M., Mäki-Arvela, P., Peixoto, A. F., Li-Zhulanov, N., Sandberg, T., Salakhutdinov, N. F., Volcho, K., Freire, C., Sidorenko, A. Y. & Murzin, D. Y., 1 Apr 2020, In: Reaction Kinetics, Mechanisms and Catalysis. 129, 2, p. 627-644 18 p.

    Research output: Contribution to journal › Article › peer-review

  77. Synthesis and analgesic activity of aliphatic ketones-derived chiral hexahydro-2H-chromenes

    Il’ina, I., Morozova, E., Pavlova, A., Korchagina, D., Tolstikova, T., Volcho, K. & Salakhutdinov, N., 1 Apr 2020, In: Medicinal Chemistry Research. 29, 4, p. 738-747 10 p.

    Research output: Contribution to journal › Article › peer-review

  78. Monoterpenoid Oximes Hydrogenation Over Platinum Catalysts

    Demidova, Y. S., Mozhaitsev, E. S., Munkuev, A. A., Suslov, E. V., Saraev, A. A., Volcho, K. P., Salakhutdinov, N. F., Simakova, I. L. & Murzin, D. Y., 1 Mar 2020, In: Topics in Catalysis. 63, 1-2, p. 187-195 9 p.

    Research output: Contribution to journal › Article › peer-review

  79. Development and validation of an LC-MS/MS method for the quantitative analysis of the anti-influenza agent camphecene in rat plasma and its application to study the blood-to-plasma distribution of the agent

    Охина, А. А., Rogachev, A. D., Yarovaya, O. I., Khvostov, M. V., Tolstikova, T. G., Покровский, А. Г., Khazanov, V. A. & Salakhutdinov, N. F., 20 Feb 2020, In: Journal of Pharmaceutical and Biomedical Analysis. 180, 11 p., 113039.

    Research output: Contribution to journal › Article › peer-review

  80. Single-stage synthesis of heterocyclic alkaloid-like compounds from (+)-camphoric acid and their antiviral activity

    Chernyshov, V. V., Yarovaya, O. I., Fadeev, D. S., Gatilov, Y. V., Esaulkova, Y. L., Muryleva, A. S., Sinegubova, K. O., Zarubaev, V. V. & Salakhutdinov, N. F., 1 Feb 2020, In: Molecular Diversity. 24, 1, p. 61-67 7 p.

    Research output: Contribution to journal › Article › peer-review

  81. Identification of novel inhibitors for the tyrosyl-DNA-phosphodiesterase 1 (Tdp1) mutant SCAN1 using virtual screening

    Mamontova, E. M., Zakharenko, A. L., Zakharova, O. D., Dyrkheeva, N. S., Volcho, K. P., Reynisson, J., Arabshahi, H. J., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jan 2020, In: Bioorganic and Medicinal Chemistry. 28, 1, 11 p., 115234.

    Research output: Contribution to journal › Article › peer-review

  82. Promising new inhibitors of tyrosyl-DNA phosphodiesterase I (Tdp 1) combining 4- arylcoumarin and monoterpenoid moieties as components of complex antitumor therapy

    Khomenko, T. M., Zakharenko, A. L., Chepanova, A. A., Ilina, E. S., Zakharova, O. D., Kaledin, V. I., Nikolin, V. P., Popova, N. A., Korchagina, D. V., Reynisson, J., Chand, R., Ayine-tora, D. M., Patel, J., Leung, I. K. H., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jan 2020, In: International Journal of Molecular Sciences. 21, 1, 21 p., 126.

    Research output: Contribution to journal › Article › peer-review

  83. Synthesis and analgesic activity of monoterpenoid aldehyde-derived hydro-2H-chromeneols

    Il'ina, I., Morozova, E., Korсhagina, D., Volсho, K., Tolstikova, T. & Salakhutdinov, N., 1 Jan 2020, In: Letters in Drug Design and Discovery. 17, 1, p. 68-78 11 p.

    Research output: Contribution to journal › Article › peer-review

  84. Modulators of Hematopoiesis Disorders (a Review)

    Salakhutdinov, N. F., Laev, S. S. & Sergeevichev, D. S., 2020, In: Chemistry for Sustainable Development. 28, 4, p. 332-353 22 p.

    Research output: Contribution to journal › Review article › peer-review

  85. 2019

  86. Clay nanotubes catalyzed solvent-free synthesis of octahydro-2H-chromenols with pharmaceutical potential from (-)-isopulegol and ketones

    Sidorenko, A. Y., Kravtsova, A. V., Il'ina, I. V., Wärnå, J., Korchagina, D. V., Gatilov, Y. V., Volcho, K. P., Salakhutdinov, N. F., Murzin, D. Y. & Agabekov, V. E., 1 Dec 2019, In: Journal of Catalysis. 380, p. 145-152 8 p.

    Research output: Contribution to journal › Article › peer-review

  87. One-Pot Myrtenol Amination over Au, Au–Pd and Pd Nanoparticles Supported on Alumina

    Demidova, Y. S., Simakova, I. L., Estrada, M., Beloshapkin, S., Suslov, E. V., Volcho, K. P., Salakhutdinov, N. F., Simakov, A. & Murzin, D. Y., 1 Dec 2019, In: Catalysis Letters. 149, 12, p. 3454-3464 11 p.

    Research output: Contribution to journal › Article › peer-review

  88. Synthesis and structure-activity relationships of novel camphecene analogues as anti-influenza agents

    Yarovaya, O. I., Sokolova, A. S., Mainagashev, I. Y., Volobueva, A. S., Lantseva, K., Borisevich, S. S., Shtro, A. A., Zarubaev, V. V. & Salakhutdinov, N. F., 1 Dec 2019, In: Bioorganic and Medicinal Chemistry Letters. 29, 23, 126745.

    Research output: Contribution to journal › Article › peer-review

  89. The first example of the stereoselective synthesis and crystal structure of a spirobicycloquinazolinone based on (-)-fenchone and anthranilamide

    Chernyshov, V. V., Gatilov, Y. V., Yarovaya, O. I., Koskin, I. P., Yarovoy, S. S., Brylev, K. A. & Salakhutdinov, N. F., 1 Dec 2019, In: Acta Crystallographica Section C: Structural Chemistry. 75, p. 1675-1680 6 p.

    Research output: Contribution to journal › Article › peer-review

  90. Comparison of dried matrix spots and fabric phase sorptive extraction methods for quantification of highly potent analgesic activity agent (2R,4aR,7R,8aR)-4,7-dimethyl-2-(thiophen-2-yl)octahydro-2H-chromen-4-ol in rat whole blood and plasma using LC–MS/MS

    Lastovka, A. V., Rogachev, A. D., Il'ina, I. V., Kabir, A., Volcho, K. P., Fadeeva, V. P., Pokrovsky, A. G., Furton, K. G. & Salakhutdinov, N. F., 15 Nov 2019, In: Journal of Chromatography B: Analytical Technologies in the Biomedical and Life Sciences. 1132, 121813.

    Research output: Contribution to journal › Article › peer-review

  91. Effective Inhibitors of Tyrosyl-DNA Phosphodiesterase 1 Based on Monoterpenoids as Potential Agents for Antitumor Therapy

    Chepanova, A. A., Li-Zhulanov, N. S., Sukhikh, A. S., Zafar, A., Reynisson, J., Zakharenko, A. L., Zakharova, O. D., Korchagina, D. V., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Nov 2019, In: Russian Journal of Bioorganic Chemistry. 45, 6, p. 647-655 9 p.

    Research output: Contribution to journal › Article › peer-review

  92. Prins cyclization of (-)-isopulegol with benzaldehyde for production of chromenols over organosulfonic clays

    Li-Zhulanov, N., Mäki-Arvela, P., Laluc, M., Peixoto, A. F., Kholkina, E., Sandberg, T., Aho, A., Volcho, K., Salakhutdinov, N., Freire, C., Sidorenko, A. Y. & Murzin, D. Y., 1 Nov 2019, In: Molecular Catalysis. 478, 12 p., 110569.

    Research output: Contribution to journal › Article › peer-review

  93. Studying Dependences Between the Chemotype Structure of Some Natural Compounds and the Spectrum of Their Targeted Activities Correlated with the Hypoglycemic Effect

    Vasilyev, P. M., Luzina, O. A., Babkov, D. A., Appazova, D. T., Salakhutdinov, N. F. & Spasov, A. A., 1 Nov 2019, In: Journal of Structural Chemistry. 60, 11, p. 1827-1832 6 p.

    Research output: Contribution to journal › Article › peer-review

  94. Synthesis of Camphecene and Cytisine Conjugates Using Click Chemistry Methodology and Study of Their Antiviral Activity

    Artyushin, O. I., Moiseeva, A. A., Zarubaev, V. V., Slita, A. V., Galochkina, A. V., Muryleva, A. A., Borisevich, S. S., Yarovaya, O. I., Salakhutdinov, N. F. & Brel, V. K., 29 Oct 2019, In: Chemistry and Biodiversity. 16, 11, e1900340.

    Research output: Contribution to journal › Article › peer-review

  95. A Novel Small Molecule Supports the Survival of Cultured Dopamine Neurons and May Restore the Dopaminergic Innervation of the Brain in the MPTP Mouse Model of Parkinson's Disease

    Ardashov, O. V., Pavlova, A. V., Mahato, A. K., Sidorova, Y., Morozova, E. A., Korchagina, D. V., Salnikov, G. E., Genaev, A. M., Patrusheva, O. S., Li-Zhulanov, N. S., Tolstikova, T. G., Volcho, K. P. & Salakhutdinov, N. F., 16 Oct 2019, In: ACS chemical neuroscience. 10, 10, p. 4337-4349 25 p.

    Research output: Contribution to journal › Article › peer-review

  96. New hydrazinothiazole derivatives of usnic acid as potent TDP1 inhibitors

    Filimonov, A. S., Chepanova, A. A., Luzina, O. A., Zakharenko, A. L., Zakharova, O. D., Ilina, E. S., Dyrkheeva, N. S., Kuprushkin, M. S., Kolotaev, A. V., Khachatryan, D. S., Patel, J., Leung, I. K. H., Chand, R., Ayine-Tora, D. M., Reynisson, J., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 15 Oct 2019, In: Molecules. 24, 20, 3711.

    Research output: Contribution to journal › Article › peer-review

  97. Dehydroabietylamine Ureas and Thioureas as Tyrosyl-DNA Phosphodiesterase 1 Inhibitors That Enhance the Antitumor Effect of Temozolomide on Glioblastoma Cells

    Kovaleva, K., Oleshko, O., Mamontova, E., Yarovaya, O., Zakharova, O., Zakharenko, A., Kononova, A., Dyrkheeva, N., Cheresiz, S., Pokrovsky, A., Lavrik, O. & Salakhutdinov, N., 27 Sept 2019, In: Journal of Natural Products. 82, 9, p. 2443-2450 8 p.

    Research output: Contribution to journal › Article › peer-review

  98. Synthesis and Hypoglycemic Activity of Aryl(Hetaryl)Propenoic Cyanopyrrolidine Amides

    Kuranov, S. O., Blokhin, M. E., Borisov, S. A., Khvostov, M. V., Luzina, O. A. & Salakhutdinov, N. F., 1 Sept 2019, In: Russian Journal of Bioorganic Chemistry. 45, 5, p. 374-380 7 p.

    Research output: Contribution to journal › Article › peer-review

  99. 1-Адамантил-3-(((1R,4aS,10aR)-7-изопропил-1,4а-диметил-1,2,3,4,4а,9,10,10а-октагидрофенантрен-1-ил)метил)мочевина, проявляющая ингибирующее действие в отношении фермента тирозил-ДНК-фосфодиэстеразы 1 человека и увеличивающая активность темозоломида в отношении клеток глиобластомы

    Олешко, О. С., Ковалева, К. С., Яровая, О. И., Мамонтова, Е. М., Захаренко, А. Л., Захарова, О. Д., Чересиз, С. В., Покровский, А. Г., Лаврик, О. И. & Салахутдинов, Н. Ф., 14 Aug 2019, IPC No. C07C275/22, C07C275/24, A61K31/17, A61P35/00, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2697409, Priority date 30 Apr 2019, Priority No. 2019113591

    Research output: Patent › Patent for invention

  100. Antimicrobial Activity of Substituted Benzopentathiepin-6-amines

    Khomenko, T. M., Korchagina, D. V., Baev, D. S., Vassiliev, P. M., Volcho, K. P. & Salakhutdinov, N. F., 1 Aug 2019, In: Journal of Antibiotics. 72, 8, p. 590-599 10 p.

    Research output: Contribution to journal › Article › peer-review

  101. Novel derivatives of deoxycholic acid bearing linear aliphatic diamine and aminoalcohol moieties and their cyclic analogs at the C3 position: Synthesis and evaluation of their in vitro antitumor potential

    Markov, A. V., Babich, V. O., Popadyuk, I. I., Salomatina, O. V., Logashenko, E. B., Salakhutdinov, N. F. & Zenkova, M. A., 21 Jul 2019, In: Molecules. 24, 14, 19 p., 2644;.

    Research output: Contribution to journal › Article › peer-review

  102. Complexes of Zn(II) and Сu(II) with the Amino Derivatives of Deoxycholic Acid: Syntheses, Structures, and Properties

    Kokina, T. E., Salomatina, O. V., Popadyuk, I. I., Glinskaya, L. A., Korol’kov, I. V., Sheludyakova, L. A., Rakhmanova, M. I. & Salakhutdinov, N. F., 1 Jul 2019, In: Russian Journal of Coordination Chemistry/Koordinatsionnaya Khimiya. 45, 7, p. 505-511 7 p.

    Research output: Contribution to journal › Article › peer-review

  103. The development of Tyrosyl-DNA phosphodiesterase 1 inhibitors. Combination of Monoterpene and Adamantine Moieties via Amide or Thioamide Bridges

    Chepanova, A. A., Mozhaitsev, E. S., Munkuev, A. A., Suslov, E. V., Korchagina, D. V., Zakharova, O. D., Zakharenko, A. L., Patel, J., Ayine-Tora, D. M., Reynisson, J., Leung, I. K. H., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jul 2019, In: Applied Sciences (Switzerland). 9, 13, 2767.

    Research output: Contribution to journal › Article › peer-review

  104. Highly selective Prins reaction over acid-modified halloysite nanotubes for synthesis of isopulegol-derived 2H-chromene compounds

    Sidorenko, A. Y., Kravtsova, A. V., Aho, A., Heinmaa, I., Wärnå, J., Pazniak, H., Volcho, K. P., Salakhutdinov, N. F., Murzin, D. Y. & Agabekov, V. E., 1 Jun 2019, In: Journal of Catalysis. 374, p. 360-377 18 p.

    Research output: Contribution to journal › Article › peer-review

  105. Synthesis and analgesic activity of octahydro-2H-chromenols, derivatives of aliphatic ketones

    Il’ina, I. V., Korchagina, D. V., Morozova, E. A., Tolstikova, T. G., Volcho, K. P. & Salakhutdinov, N. F., 1 May 2019, In: Russian Chemical Bulletin. 68, 5, p. 1061-1066 6 p.

    Research output: Contribution to journal › Article › peer-review

  106. Synthesis, hypolipidemic and antifungal activity of tetrahydroberberrubine sulfonates

    Nechepurenko, I. V., Shirokova, E. D., Khvostov, M. V., Frolova, T. S., Sinitsyna, O. I., Maksimov, A. M., Bredikhin, R. A., Komarova, N. I., Fadeev, D. S., Luzina, O. A., Tolstikova, T. G. & Salakhutdinova, N. F., 1 May 2019, In: Russian Chemical Bulletin. 68, 5, p. 1052-1060 9 p.

    Research output: Contribution to journal › Article › peer-review

  107. Synthesis of (1S)-(+)-camphor-10-sulfonic acid derivatives and investigations in vitro and in silico of their antiviral activity as the inhibitors of fi lovirus infections

    Sokolova, A. S., Baranova, D. V., Yarovaya, O. I., Baev, D. S., Polezhaeva, O. A., Zybkina, A. V., Shcherbakov, D. N., Tolstikova, T. G. & Salakhutdinov, N. F., 1 May 2019, In: Russian Chemical Bulletin. 68, 5, p. 1041-1046 6 p.

    Research output: Contribution to journal › Article › peer-review

  108. Effect of chiral polyhydrochromenes on cannabinoid system

    Li-Zhulanov, N. S., Il’ina, I. V., Chicca, A., Schenker, P., Patrusheva, O. S., Nazimova, E. V., Korchagina, D. V., Krasavin, M., Volcho, K. P. & Salakhutdinov, N. F., Apr 2019, In: Medicinal Chemistry Research. 28, 4, p. 450-464 15 p.

    Research output: Contribution to journal › Article › peer-review

  109. Antimetastatic Activity of Combined Topotecan and Tyrosyl-DNA Phosphodiesterase-1 Inhibitor on Modeled Lewis Lung Carcinoma

    Koldysheva, E. V., Men’shchikova, A. P., Lushnikova, E. L., Popova, N. A., Kaledin, V. I., Nikolin, V. P., Zakharenko, A. L., Luzina, O. A., Salakhutdinov, N. F. & Lavrik, O. I., 15 Mar 2019, In: Bulletin of Experimental Biology and Medicine. 166, 5, p. 661-666 6 p.

    Research output: Contribution to journal › Article › peer-review

  110. Synthesis of diazaadamantanes from 1,5-dimethylbispidinone and some natural ketones

    Suslov, E. V., Ponomarev, K. Y., Korchagina, D. V., Volcho, K. P. & Salakhutdinov, N. F., 1 Mar 2019, In: Russian Chemical Bulletin. 68, 3, p. 601-605 5 p.

    Research output: Contribution to journal › Article › peer-review

  111. Increasing bioavailability of very poorly water-soluble compounds. A case study of an anti-tumor drug, soloxolon methyl

    Ogienko, A. G., Markov, A. V., Sen'kova, A. V., Logashenko, E. B., Salomatina, O. V., Myz, S. A., Ogienko, A. A., Nefedov, A. A., Losev, E. A., Drebushchak, T. N., Salakhutdinov, N. F., Boldyrev, V. V., Vlasov, V. V., Zenkova, M. A. & Boldyreva, E. V., 1 Feb 2019, In: Journal of Drug Delivery Science and Technology. 49, p. 35-42 8 p.

    Research output: Contribution to journal › Article › peer-review

  112. Inhibitory Effect of New Semisynthetic Usnic Acid Derivatives on Human Tyrosyl-DNA Phosphodiesterase 1

    Dyrkheeva, N., Luzina, O., Filimonov, A., Zakharova, O., Ilina, E., Zakharenko, A., Kuprushkin, M., Nilov, D., Gushchina, I., Švedas, V., Salakhutdinov, N. & Lavrik, O., 1 Jan 2019, In: Planta Medica. 85, 2, p. 103-111 9 p.

    Research output: Contribution to journal › Article › peer-review

  113. Neuroregeneration in Parkinson's Disease: From Proteins to Small Molecules

    Sidorova, Y. A., Volcho, K. P. & Salakhutdinov, N. F., 1 Jan 2019, In: Current Neuropharmacology. 17, 3, p. 268-287 20 p.

    Research output: Contribution to journal › Review article › peer-review

  114. Novel inhibitors of DNA repair enzyme TDP1 combining monoterpenoid and adamantane fragments

    Mozhaitsev, E. S., Zakharenko, A. L., Suslov, E. V., Korchagina, D. V., Zakharova, O. D., Vasil’eva, I. A., Chepanova, A. A., Black, E., Patel, J., Chand, R., Reynisson, J., Leung, I. K. H., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jan 2019, In: Anti-Cancer Agents in Medicinal Chemistry. 19, 4, p. 463-472 10 p.

    Research output: Contribution to journal › Article › peer-review

  115. Novel tyrosyl-DNA phosphodiesterase 1 inhibitors enhance the therapeutic impact of topoteсan on in vivo tumor models

    Zakharenko, A. L., Luzina, O. A., Sokolov, D. N., Kaledin, V. I., Nikolin, V. P., Popova, N. A., Patel, J., Zakharova, O. D., Chepanova, A. A., Zafar, A., Reynisson, J., Leung, E., Leung, I. K. H., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jan 2019, In: European Journal of Medicinal Chemistry. 161, p. 581-593 13 p.

    Research output: Contribution to journal › Article › peer-review

  116. The development of tyrosyl-DNA phosphodyesterase 1 (TDP1) inhibitors based on the amines combining aromatic/heteroaromatic and monoterpenoid moieties

    Mozhaitsev, E., Suslov, E., Demidova, Y., Korchagina, D., Volcho, K., Zakharenko, A., Vasil’eva, I., Kupryushkin, M., Chepanova, A., Ayine-Tora, D. M., Reynisson, J., Salakhutdinov, N. & Lavrik, O., 1 Jan 2019, In: Letters in Drug Design and Discovery. 16, 5, p. 597-605 9 p.

    Research output: Contribution to journal › Article › peer-review

  117. Effects of acute and chronic treatment of STEP inhibitor, TC-2153, on the nervous system and behaviour of zebrafish (Danio rerio)

    Kulikov, A., Sinyakova, N., Kulikova, E., Evglevsky, N., Kolotygin, I., Volcho, K., Salakhutdinov, N., Kulikov, V., Romaschenko, A. & Moshkin, M., 2019, In: European Neuropsychopharmacology. 29, p. S198-S199 2 p.

    Research output: Contribution to journal › Meeting Abstract › peer-review

  118. 2018

  119. Molecular and Supramolecular Structure of 8-(Trifluoromethyl)Benzo[f][1,2,3,4,5] Pentathiepin-6-Amine – A Representative of Condensed Arene Pentathiepines

    Rybalova, T. V., Rogachev, A. D., Khomenko, T. M., Volcho, K. P. & Salakhutdinov, N. F., 1 Dec 2018, In: Journal of Structural Chemistry. 59, 7, p. 1753-1758 6 p.

    Research output: Contribution to journal › Article › peer-review

  120. Synthesis of d-(+)-camphor-based: N -acylhydrazones and their antiviral activity

    Kovaleva, K. S., Zubkov, F. I., Bormotov, N. I., Novikov, R. A., Dorovatovskii, P. V., Khrustalev, V. N., Gatilov, Y. V., Zarubaev, V. V., Yarovaya, O. I., Shishkina, L. N. & Salakhutdinov, N. F., 1 Dec 2018, In: MedChemComm. 9, 12, p. 2072-2082 11 p.

    Research output: Contribution to journal › Article › peer-review

  121. Untargeted search and identification of metabolites of antiviral agent camphecene in rat urine by liquid chromatography and mass spectrometry and studying their distribution in organs following peroral administration of the compound

    Rogachev, A. D., Yarovaya, O. I., Fatianova, A. V., Lavrinenko, V. A., Amosov, E. V., Zarubaev, V. V., Pokrovsky, A. G. & Salakhutdinov, N. F., 30 Nov 2018, In: Journal of Pharmaceutical and Biomedical Analysis. 161, p. 383-392 10 p.

    Research output: Contribution to journal › Article › peer-review

  122. Preparation of chiral isobenzofurans from 3-carene in the presence of modified clays

    Sidorenko, A. Y., Il'ina, I. V., Kravtsova, A. V., Aho, A., Ardashov, O. V., Li-Zhulanov, N. S., Volcho, K. P., Salakhutdinov, N. F., Murzin, D. Y. & Agabekov, V. E., 1 Nov 2018, In: Molecular Catalysis. 459, p. 38-45 8 p.

    Research output: Contribution to journal › Article › peer-review

  123. Selection of influenza virus resistant to the novel camphor-based antiviral camphecene results in loss of pathogenicity

    Zarubaev, V. V., Pushkina, E. A., Borisevich, S. S., Galochkina, A. V., Garshinina, A. V., Shtro, A. A., Egorova, A. A., Sokolova, A. S., Khursan, S. L., Yarovaya, O. I. & Salakhutdinov, N. F., 1 Nov 2018, In: Virology. 524, p. 69-77 9 p.

    Research output: Contribution to journal › Article › peer-review

  124. Highly selective reduction of nitroarenes by sc-isopropanol in the presence of zirconia in a flow reactor

    Anikeev, V. I., Sivcev, V. P., Valeev, K. R., Volcho, K. P., Sadykov, V. A. & Salakhutdinov, N. F., 1 Oct 2018, In: Journal of Supercritical Fluids. 140, p. 233-237 5 p.

    Research output: Contribution to journal › Article › peer-review

  125. Synthesis and antiviral activity of camphor-based 1,3-thiazolidin-4-one and thiazole derivatives as Orthopoxvirus-reproduction inhibitors

    Sokolova, A. S., Yarovaya, O. I., Bormotov, N. I., Shishkina, L. N. & Salakhutdinov, N. F., 1 Oct 2018, In: MedChemComm. 9, 10, p. 1746-1753 8 p.

    Research output: Contribution to journal › Article › peer-review

  126. A novel class of tyrosyl-DNA phosphodiesterase 1 inhibitors that contains the octahydro-2H-chromen-4-ol scaffold

    Li-Zhulanov, N. S., Zakharenko, A. L., Chepanova, A. A., Patel, J., Zafar, A., Volcho, K. P., Salakhutdinov, N. F., Reynisson, J., Leung, I. K. H. & Lavrik, O. I., 26 Sept 2018, In: Molecules. 23, 10, 14 p., 2468.

    Research output: Contribution to journal › Article › peer-review

  127. Discovery of a New Class of Inhibitors of Vaccinia Virus Based on (−)-Borneol from Abies sibirica and (+)-Camphor

    Sokolova, A. S., Yarovaya, O. I., Bormotov, N. I., Shishkina, L. N. & Salakhutdinov, N. F., 1 Sept 2018, In: Chemistry and Biodiversity. 15, 9, 9 p., e1800153.

    Research output: Contribution to journal › Article › peer-review

  128. Synthesis and evaluation of aryliden- and hetarylidenfuranone derivatives of usnic acid as highly potent Tdp1 inhibitors

    Zakharova, O., Luzina, O., Zakharenko, A., Sokolov, D., Filimonov, A., Dyrkheeva, N., Chepanova, A., Ilina, E., Ilyina, A., Klabenkova, K., Chelobanov, B., Stetsenko, D., Zafar, A., Eurtivong, C., Reynisson, J., Volcho, K., Salakhutdinov, N. & Lavrik, O., 15 Aug 2018, In: Bioorganic and Medicinal Chemistry. 26, 15, p. 4470-4480 11 p.

    Research output: Contribution to journal › Article › peer-review

  129. Synthesis and evaluation of camphor and cytisine-based cyanopyrrolidines as DPP-IV inhibitors for the treatment of type 2 diabetes mellitus

    Kuranov, S. O., Tsypysheva, I. P., Khvostov, M. V., Zainullina, L. F., Borisevich, S. S., Vakhitova, Y. V., Luzina, O. A. & Salakhutdinov, N. F., 15 Aug 2018, In: Bioorganic and Medicinal Chemistry. 26, 15, p. 4402-4409 8 p.

    Research output: Contribution to journal › Article › peer-review

  130. Preparation of octahydro-2H-chromen-4-ol with analgesic activity from isopulegol and thiophene-2-carbaldehyde in the presence of acid-modified clays

    Sidorenko, A. Y., Kravtsova, A. V., Wärnå, J., Aho, A., Heinmaa, I., Il'ina, I. V., Ardashov, O. V., Volcho, K. P., Salakhutdinov, N. F., Murzin, D. Y. & Agabekov, V. E., 1 Jul 2018, In: Molecular Catalysis. 453, p. 139-148 10 p.

    Research output: Contribution to journal › Article › peer-review

  131. Synthesis and Inhibitory Properties of Imines Containing Monoterpenoid and Adamantane Fragments Against DNA Repair Enzyme Tyrosyl-DNA Phosphodiesterase 1 (Tdp1)

    Zakharenko, A. L., Mozhaitsev, E. S., Suslov, E. V., Korchagina, D. V., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jul 2018, In: Chemistry of Natural Compounds. 54, 4, p. 672-676 5 p.

    Research output: Contribution to journal › Article › peer-review

  132. Highly potent activity of isopulegol-derived substituted octahydro-2H-chromen-4-ols against influenza A and B viruses

    Ilyina, I. V., Zarubaev, V. V., Lavrentieva, I. N., Shtro, A. A., Esaulkova, I. L., Korchagina, D. V., Borisevich, S. S., Volcho, K. P. & Salakhutdinov, N. F., 15 Jun 2018, In: Bioorganic and Medicinal Chemistry Letters. 28, 11, p. 2061-2067 7 p.

    Research output: Contribution to journal › Article › peer-review

  133. Usnic acid and its derivatives for pharmaceutical use: a patent review (2000–2017)

    Luzina, O. A. & Salakhutdinov, N. F., 3 Jun 2018, In: Expert Opinion on Therapeutic Patents. 28, 6, p. 477-491 15 p.

    Research output: Contribution to journal › Review article › peer-review

  134. 3-N-ЗАМЕЩЕННЫЕ БОРНИЛПРОПИОНАТЫ, ИСПОЛЬЗУЕМЫЕ В КАЧЕСТВЕ ИНГИБИТОРОВ ВИРУСА МАРБУРГ

    Яровая, О. И., Соколова, А. С., Кононова, А. А., Чересиз, С. В., Никитина, Р. А., Чепурнов, А. А., Зайковская, А. В., Пьянков, О. В., Покровский, А. Г., Максютов, Р. А. & Салахутдинов, Н. Ф., 3 Apr 2018, IPC No. A61K31/4453, A61K31/452, A61P31/12, C07D211/14, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2649406, Priority date 21 Sept 2017, Priority No. 2017133088

    Research output: Patent › Patent for invention

  135. One-pot monoterpene alcohol amination over Au/ZrO2 catalyst: Effect of the substrate structure

    Demidova, Y. S., Suslov, E. V., Simakova, I. L., Mozhajcev, E. S., Korchagina, D. V., Volcho, K. P., Salakhutdinov, N. F., Simakov, A. & Murzin, D. Y., 1 Apr 2018, In: Journal of Catalysis. 360, p. 127-134 8 p.

    Research output: Contribution to journal › Article › peer-review

  136. Novel semisynthetic derivatives of bile acids as effective tyrosyl-DNA phosphodiesterase 1 inhibitors

    Salomatina, O. V., Popadyuk, I. I., Zakharenko, A. L., Zakharova, O. D., Fadeev, D. S., Komarova, N. I., Reynisson, J., Arabshahi, H. J., Chand, R., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 17 Mar 2018, In: Molecules. 23, 3, 19 p., 679.

    Research output: Contribution to journal › Article › peer-review

  137. Antiulcerogenic activity of borneol derivatives

    Borisova, M. S., Yarovaya, O. I., Semenova, M. D., Tolstikova, T. G. & Salakhutdinov, N. F., 1 Mar 2018, In: Russian Chemical Bulletin. 67, 3, p. 558-561 4 p.

    Research output: Contribution to journal › Article › peer-review

  138. Development and Validation of a Method for Determination of a New Effective Inhibitor of Influenza Virus H1N1 in Blood Plasma

    Sokolova, A. S., Yarovaya, O. I., Nefedov, A. A. & Salakhutdinov, N. F., Mar 2018, In: Pharmaceutical Chemistry Journal. 51, 12, p. 1102-1105 4 p.

    Research output: Contribution to journal › Article › peer-review

  139. Aminoadamantanes containing monoterpene-derived fragments as potent tyrosyl-DNA phosphodiesterase 1 inhibitors

    Ponomarev, K. Y., Suslov, E. V., Zakharenko, A. L., Zakharova, O. D., Rogachev, A. D., Korchagina, D. V., Zafar, A., Reynisson, J., Nefedov, A. A., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Feb 2018, In: Bioorganic Chemistry. 76, p. 392-399 8 p.

    Research output: Contribution to journal › Article › peer-review

  140. Application of monoterpenoids and their derivatives for treatment of neurodegenerative disorders

    Volcho, K. P., Laev, S. S., Ashraf, G. M., Aliev, G. & Salakhutdinov, N. F., 1 Jan 2018, In: Current Medicinal Chemistry. 25, 39, p. 5327-5346 20 p.

    Research output: Contribution to journal › Review article › peer-review

  141. Synthesis of Sulfones and Sulfoxides Based on (+)-usnic Acid

    Sokolov, D. N., Luzina, O. A. & Salakhutdinov, N. F., 1 Jan 2018, In: Chemistry of Natural Compounds. 54, 1, p. 46-49 4 p.

    Research output: Contribution to journal › Article › peer-review

  142. 2017

  143. N-Heterocyclic borneol derivatives as inhibitors of Marburg virus glycoprotein-mediated VSIV pseudotype entry

    Kononova, A. A., Sokolova, A. S., Cheresiz, S. V., Yarovaya, O. I., Nikitina, R. A., Chepurnov, A. A., Pokrovsky, A. G. & Salakhutdinov, N. F., 1 Dec 2017, In: MedChemComm. 8, 12, p. 2233-2237 5 p.

    Research output: Contribution to journal › Article › peer-review

  144. Synthesis and analgesic activity of amines combining diazaadamantane and monoterpene fragments

    Ponomarev, K., Morozova, E., Pavlova, A., Suslov, E., Korchagina, D., Nefedov, A., Tolstikova, T., Volcho, K. & Salakhutdinov, N., 1 Dec 2017, In: Medicinal Chemistry. 13, 8, p. 773-779 7 p.

    Research output: Contribution to journal › Article › peer-review

  145. Evolution of anti-parkinsonian activity of monoterpenoid (1R,2R,6S)-3-methyl-6-(prop-1-en-2-yl)cyclohex-3-ene-1,2-diol in various in vivo models

    Valdman, E., Kapitsa, I., Ivanova, Е., Voronina, T., Ardashov, O., Volcho, K., Khazanov, V. & Salakhutdinov, N., 15 Nov 2017, In: European Journal of Pharmacology. 815, p. 351-363 13 p.

    Research output: Contribution to journal › Article › peer-review

  146. Synthesis and Analgesic Activity of 4,7-Dimethyl-3,4,4a,5,8,8a-Hexahydro-2-Chromen-4,8-Diols Containing Alkyl-Substituted Aromatic Moieties

    Patrusheva, O. S., Pavlova, A. V., Korchagina, D. V., Tolstikova, T. G., Volcho, K. P. & Salakhutdinov, N. F., 1 Nov 2017, In: Chemistry of Natural Compounds. 53, 6, p. 1066-1071 6 p.

    Research output: Contribution to journal › Article › peer-review

  147. Synthesis and Analgesic Activity of 5,7- and 6-Substituted Diazaadamantanes Containing Monoterpene Moieties

    Ponomarev, K. Y., Morozova, E. A., Suslov, E. V., Korchagina, D. V., Tolstikova, T. G., Volcho, K. P. & Salakhutdinov, N. F., 1 Nov 2017, In: Chemistry of Natural Compounds. 53, 6, p. 1131-1136 6 p.

    Research output: Contribution to journal › Article › peer-review

  148. Synthesis and evaluation of antitumor, anti-inflammatory and analgesic activity of novel deoxycholic acid derivatives bearing aryl- or hetarylsulfanyl moieties at the C-3 position

    Popadyuk, I. I., Markov, A. V., Morozova, E. A., Babich, V. O., Salomatina, O. V., Logashenko, E. B., Zenkova, M. A., Tolstikova, T. G. & Salakhutdinov, N. F., Nov 2017, In: Steroids. 127, p. 1-12 12 p.

    Research output: Contribution to journal › Article › peer-review

  149. Anti-influenza activity of diazaadamantanes combined with monoterpene moieties

    Suslov, E., Zarubaev, V. V., Slita, A. V., Ponomarev, K., Korchagina, D., Ayine-Tora, D. M., Reynisson, J., Volcho, K. & Salakhutdinov, N., 1 Oct 2017, In: Bioorganic and Medicinal Chemistry Letters. 27, 19, p. 4531-4535 5 p.

    Research output: Contribution to journal › Article › peer-review

  150. Novel derivatives of deoxycholic acid bearing aliphatic or cyclic diamine moieties at the C-3 position: Synthesis and evaluation of anti-proliferative activity

    Popadyuk, I. I., Markov, A. V., Babich, V. O., Salomatina, O. V., Logashenko, E. B., Zenkova, M. A. & Salakhutdinov, N. F., 15 Aug 2017, In: Bioorganic and Medicinal Chemistry Letters. 27, 16, p. 3755-3759 5 p.

    Research output: Contribution to journal › Article › peer-review

  151. Benzopentathiepine derivative, 8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amine hydrochloride (TC-2153), as a promising antidepressant of new generation

    Kulikova, E. A., Volcho, K. P., Salakhutdinov, N. F. & Kulikov, A. V., 1 Aug 2017, In: Letters in Drug Design and Discovery. 14, 8, p. 974-984 11 p.

    Research output: Contribution to journal › Review article › peer-review

  152. Synthesis and analgesic activity of monoterpenoid-derived alkyl-substituted chiral hexahydro-2H-chromenes

    Il’ina, I., Pavlova, A., Korchagina, D., Ardashov, O., Tolstikova, T., Volcho, K. & Salakhutdinov, N., 1 Jul 2017, In: Medicinal Chemistry Research. 26, 7, p. 1415-1426 12 p.

    Research output: Contribution to journal › Article › peer-review

  153. Synthesis of camphecene derivatives using click chemistry methodology and study of their antiviral activity

    Artyushin, O. I., Sharova, E. V., Vinogradova, N. M., Genkina, G. K., Moiseeva, A. A., Klemenkova, Z. S., Orshanskaya, I. R., Shtro, A. A., Kadyrova, R. A., Zarubaev, V. V., Yarovaya, O. I., Salakhutdinov, N. F. & Brel, V. K., 15 May 2017, In: Bioorganic and Medicinal Chemistry Letters. 27, 10, p. 2181-2184 4 p.

    Research output: Contribution to journal › Article › peer-review

  154. One-pot synthesis of 1,5,3-oxathiazepanes via the three-component condensation of primary amines, formaldehyde and 2-mercaptoethanol

    Kovaleva, K. S., Yarovaya, O. I., Fadeev, D. S. & Salakhutdinov, N. F., 10 May 2017, In: Tetrahedron Letters. 58, 19, p. 1868-1870 3 p.

    Research output: Contribution to journal › Article › peer-review

  155. Inhibitors of nuclease and redox activity of apurinic/apyrimidinic endonuclease 1/redox effector factor 1 (APE1/Ref-1)

    Laev, S. S., Salakhutdinov, N. F. & Lavrik, O. I., 1 May 2017, In: Bioorganic and Medicinal Chemistry. 25, 9, p. 2531-2544 14 p.

    Research output: Contribution to journal › Review article › peer-review

  156. Synthesis and in vitro study of novel borneol derivatives as potent inhibitors of the influenza A virus

    Sokolova, A. S., Yarovaya, O. I., Semenova, M. D., Shtro, A. A., Orshanskaya, I. R., Zarubaev, V. V. & Salakhutdinov, N. F., 1 May 2017, In: MedChemComm. 8, 5, p. 960-963 4 p.

    Research output: Contribution to journal › Article › peer-review

  157. The decisive role of mutual arrangement of hydroxy and methoxy groups in (3(4)-hydroxy-4(3)-methoxyphenyl)-4,7-dimethyl-3,4,4a,5,8,8ahexahydro- 2H-chromene-4,8-diols in their Biological Activity

    Pavlova, A., Patrusheva, O., Il'ina, I., Volcho, K., Tolstikova, T. & Salakhutdinov, N., 1 May 2017, In: Letters in Drug Design and Discovery. 14, 5, p. 508-514 7 p.

    Research output: Contribution to journal › Article › peer-review

  158. Promoting effect of alcohols and formic acid on Au-catalyzed one-pot myrtenol amination

    Demidova, Y. S., Suslov, E. V., Simakova, I. L., Volcho, K. P., Smolentseva, E., Salakhutdinov, N. F., Simakov, A. & Murzin, D. Y., May 2017, In: Molecular Catalysis. 433, p. 414-419 6 p.

    Research output: Contribution to journal › Article › peer-review

  159. Influenza Antiviral Activity of Br-Containing [2R,4R(S),4aR,7R,8aR]-4,7-Dimethyl-2-(Thiophen-2-YL)Octahydro-2H-Chromen-4-Ols Prepared from (–)-Isopulegol

    Nazimova, E. V., Shtro, A. A., Anikin, V. B., Patrusheva, O. S., Il′ina, I. V., Korchagina, D. V., Zarubaev, V. V., Volcho, K. P. & Salakhutdinov, N. F., 1 Mar 2017, In: Chemistry of Natural Compounds. 53, 2, p. 260-264 5 p.

    Research output: Contribution to journal › Article › peer-review

  160. Synthesis and biological activity of heterocyclic borneol derivatives

    Sokolova, A. S., Yarovaya, О. I., Shtro, A. A., Borisova, M. S., Morozova, E. A., Tolstikova, T. G., Zarubaev, V. V. & Salakhutdinov, N. F., 1 Mar 2017, In: Chemistry of Heterocyclic Compounds. 53, 3, p. 371-377 7 p.

    Research output: Contribution to journal › Article › peer-review

  161. Synthesis of new heterocyclic dehydroabietylamine derivatives and their biological activity

    Kovaleva, K. S., Yarovaya, O. I., Shernyukov, A. V., Zarubaev, V. V., Shtro, A. A., Orshanskaya, Y. R. & Salakhutdinov, N. F., 1 Mar 2017, In: Chemistry of Heterocyclic Compounds. 53, 3, p. 364-370 7 p.

    Research output: Contribution to journal › Article › peer-review

  162. Aliphatic and alicyclic camphor imines as effective inhibitors of influenza virus H1N1

    Sokolova, A. S., Yarovaya, О. I., Baev, D. S., Shernyukov, А. V., Shtro, A. A., Zarubaev, V. V. & Salakhutdinov, N. F., 15 Feb 2017, In: European Journal of Medicinal Chemistry. 127, p. 661-670 10 p.

    Research output: Contribution to journal › Article › peer-review

  163. Cytotoxic and cancer preventive activity of benzotrithioles and benzotrithiole oxides, synthetic analogues of varacins

    Kuzmich, A. S., Khomenko, T. M., Fedorov, S. N., Makarieva, T. N., Shubina, L. K., Komarova, N. I., Korchagina, D. V., Rybalova, T. V., Volcho, K. P. & Salakhutdinov, N. F., 1 Feb 2017, In: Medicinal Chemistry Research. 26, 2, p. 397-404 8 p.

    Research output: Contribution to journal › Article › peer-review

  164. Effect of New Antiviral Agent Camphecin on Behavior of Mice

    Babina, A. V., Lavrinenko, V. A., Yarovaya, O. I. & Salakhutdinov, N. F., 1 Jan 2017, In: Bulletin of Experimental Biology and Medicine. 162, 3, p. 346-348 3 p.

    Research output: Contribution to journal › Article › peer-review

  165. Gold catalyzed one-pot myrtenol amination: Effect of catalyst redox activation

    Simakova, I. L., Demidova, Y. S., Estrada, M., Beloshapkin, S., Suslov, E. V., Volcho, K. P., Salakhutdinov, N. F., Murzin, D. Y. & Simakov, A., 1 Jan 2017, In: Catalysis Today. 279, p. 63-70 8 p.

    Research output: Contribution to journal › Article › peer-review

  166. Selectivity control in one-pot myrtenol amination over Au/ZrO2 by molecular hydrogen addition

    Demidova, Y. S., Suslov, E. V., Simakova, I. L., Mozhajcev, E. S., Korchagina, D. V., Volcho, K. P., Salakhutdinov, N. F., Simakov, A. & Murzin, D. Y., 1 Jan 2017, In: Journal of Molecular Catalysis A: Chemical. 426, p. 60-67 8 p.

    Research output: Contribution to journal › Article › peer-review

  167. Two-step synthesis of monoterpenoid dioxinols exhibiting analgesic activity from isopulegol and benzaldehyde over heterogeneous catalysts

    Stekrova, M., Mäki-Arvela, P., Leino, E., Valkaj, K. M., Eränen, K., Aho, A., Smeds, A., Kumar, N., Volcho, K. P., Salakhutdinov, N. F. & Murzin, D. Y., 1 Jan 2017, In: Catalysis Today. 279, p. 56-62 7 p.

    Research output: Contribution to journal › Article › peer-review

  168. Usnic acid derivatives are effective inhibitors of tyrosyl-DNA phosphodiesterase 1

    Zakharenko, A. L., Luzina, O. A., Sokolov, D. N., Zakharova, O. D., Rakhmanova, M. E., Chepanova, A. A., Dyrkheeva, N. S., Lavrik, O. I. & Salakhutdinov, N. F., 1 Jan 2017, In: Russian Journal of Bioorganic Chemistry. 43, 1, p. 84-90 7 p.

    Research output: Contribution to journal › Article › peer-review

  169. Anti-influenza activity of monoterpene-containing substituted coumarins

    Khomenko, T. M., Zarubaev, V. V., Orshanskaya, I. R., Kadyrova, R. A., Sannikova, V. A., Korchagina, D. V., Volcho, K. P. & Salakhutdinov, N. F., 2017, In: Bioorganic and Medicinal Chemistry Letters. 27, 13, p. 2920-2925 6 p.

    Research output: Contribution to journal › Article › peer-review

  170. Modern approaches to modification of bile acids for the synthesis of compounds possessing valuable physicochemical and biological properties

    Popadyuk, I. I., Salomatina, O. V. & Salakhutdinov, N. F., 2017, In: Russian Chemical Reviews. 86, 5, p. 388-443 56 p.

    Research output: Contribution to journal › Review article › peer-review

  171. 2016

  172. Development and validation of ultrafast LC–MS/MS method for quantification of anti-influenza agent camphecene in whole rat blood using dried blood spots and its application to pharmacokinetic studies

    Rogachev, A. D., Yarovaya, O. I., Ankov, S. V., Khvostov, M. V., Tolstikova, T. G., Pokrovsky, A. G. & Salakhutdinov, N. F., 15 Nov 2016, In: Journal of Chromatography B: Analytical Technologies in the Biomedical and Life Sciences. 1036-1037, p. 136-141 6 p.

    Research output: Contribution to journal › Article › peer-review

  173. Chemical approach to the design of effective antidiabetic agents

    Rogachev, A. D., Kuranov, S. O. & Salakhutdinov, N. F., 2016, In: Russian Chemical Reviews. 85, 12, p. 1313-1337 25 p.

    Research output: Contribution to journal › Review article › peer-review

  174. 2015

  175. Synthesis and analgesic activity of stereoisomers of 2-(3(4)-hydroxy-4(3)-methoxyphenyl)-4,7-dimethyl-3,4,4a,5,8,8a-hexahydro-2H-chromene-4,8-diols

    Pavlova, A., Mikhalchenko, O., Rogachev, A., Il'ina, I., Korchagina, D., Gatilov, Y., Tolstikova, T., Volcho, K. & Salakhutdinov, N., 28 Nov 2015, In: Medicinal Chemistry Research. 24, 11, p. 3821-3830 10 p.

    Research output: Contribution to journal › Article › peer-review

  176. Compounds combining aminoadamantane and monoterpene moieties: Cytotoxicity and mutagenic effects

    Suslov, E. V., Ponomarev, K. Y., Rogachev, A. D., Pokrovsky, M. A., Pokrovsky, A. G., Pykhtina, M. B., Beklemishev, A. B., Korchagina, D. V., Volcho, K. P. & Salakhutdinov, N. F., 1 Oct 2015, In: Medicinal Chemistry. 11, 7, p. 629-635 7 p.

    Research output: Contribution to journal › Article › peer-review

  177. Unique shortening of carbon chain during reduction of aliphatic nitro compounds to amines in the presence of supercritical isopropanol on alumina

    Sivcev, V. P., Volcho, K. P., Salakhutdinov, N. F. & Anikeev, V. I., 28 Jul 2015, In: Journal of Supercritical Fluids. 103

    Research output: Contribution to journal › Article › peer-review

  178. Isomerization of verbenol oxide to a diol with para-menthane structure exhibiting anti-Parkinson activity

    Torozova, A., Mäki-Arvela, P., Kumar, N., Aho, A., Smeds, A., Peurla, M., Sjöholm, R., Heinmaa, I., Volcho, K. P., Salakhutdinov, N. F. & Murzin, D. Y., 24 Jul 2015, In: Reaction Kinetics, Mechanisms and Catalysis. 116, 2

    Research output: Contribution to journal › Article › peer-review

  179. Chemical Composition of Pinus sibirica (Pinaceae)

    Rogachev, A. D. & Salakhutdinov, N. F., Jan 2015, In: Chemistry and Biodiversity. 12, 1, p. 1-53 53 p.

    Research output: Contribution to journal › Review article › peer-review

  180. 2014

  181. ПРОИЗВОДНЫЕ УСНИНОВОЙ КИСЛОТЫ КАК ПРОТИВООПУХОЛЕВЫЕ АГЕНТЫ

    Покровский, А. Г., Покровский, М. А., Лузина, О. А., Соколов, Д. Н. & Салахутдинов, Н. Ф., 27 Dec 2014, IPC No. C07D493/04, A61K31/343, A61K35/00, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2536873, Priority date 30 Sept 2013, Priority No. 2013143977

    Research output: Patent › Patent for invention

  182. 4-ИЗОПРОПИЛ-7-МЕТОКСИ-2А1-МЕТИЛ-2,2А,2А1,3,5А,9B-ГЕКСАГИДРОФЛУОРЕНО[9,1-BC]ФУРАН-8-ОЛ, ОБЛАДАЮЩИЙ ПРОТИВООПУХОЛЕВОЙ АКТИВНОСТЬЮ

    Покровский, А. Г., Покровский, М. А., Курбакова, С. Ю., Корчагина, Д. В., Михальченко, О. С., Волчо, К. П. & Салахутдинов, Н. Ф., 20 Dec 2014, IPC No. C07D307/77, A61K31/343, A61P35/00, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2535926, Priority date 30 Sept 2013, Priority No. 2013143979

    Research output: Patent › Patent for invention

  183. 2013

  184. Synthesis of new compounds combining adamantanamine and monoterpene fragments and their antiviral activity against influenza virus A(H1N1)pdm09

    Teplov, G. V., Suslov, E. V., Zarubaev, V. V., Shtro, A. A., Karpinskaya, L. A., Rogachev, A. D., Korchagina, D. V., Volcho, K. P., Salakhutdinov, N. F. & Kiselev, O. I., Jul 2013, In: Letters in Drug Design and Discovery. 10, 6, p. 477-485 9 p.

    Research output: Contribution to journal › Article › peer-review

  185. Aryloxyacetamides derived from resveratroloside and pinostilbenoside

    Pozdeeva, A. V., Komarova, N. I., Vasiliev, V. G., Rogachev, A. D., Salakhutdinov, N. F. & Tolstikov, G. A., Jan 2013, In: Mendeleev Communications. 23, 1, p. 37-38 2 p.

    Research output: Contribution to journal › Article › peer-review

  186. 2012

  187. ГИДРИРОВАННАЯ БЕТУЛОНОВАЯ КИСЛОТА И ЕЕ АМИДЫ КАК ПРОТИВООПУХОЛЕВЫЕ СРЕДСТВА ТРИТЕРПЕНОВОЙ ПРИРОДЫ

    Покровский, А. Г., Покровский, М. А., Салахутдинов, Н. Ф., Толстиков, Г. А. & Майнагашев, И. Я., 20 Apr 2012, IPC No. C07J53/00, C07J63/00, A61P35/00, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2448115, Priority date 20 Dec 2010, Priority No. 2010152163

    Research output: Patent › Patent for invention

  188. N-ЭТИЛПИПЕРАЗИЛАМИД БЕТУЛОНОВОЙ КИСЛОТЫ КАК ПРОТИВООПУХОЛЕВОЕ СРЕДСТВО ТРИТЕРПЕНОВОЙ ПРИРОДЫ

    Покровский, А. Г., Покровский, М. А., Салахутдинов, Н. Ф., Толстиков, Г. А. & Майнагашев, И. Я., 20 Mar 2012, IPC No. C07J53/00, C07J43/00, A61P35/00, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2445317, Priority date 28 Oct 2010, Priority No. 2010144219

    Research output: Patent › Patent for invention

  189. Reaction of several resveratrol glycoside derivatives with hypochlorites in various media

    Rogachev, A. D., Komarova, N. I., Pozdeeva, A. V., Korchagina, D. V., Vasil'Ev, V. G., Salakhutdinov, N. F. & Tolstikov, G. A., Mar 2012, In: Chemistry of Natural Compounds. 48, 1, p. 1-7 7 p.

    Research output: Contribution to journal › Article › peer-review

  190. 2009

  191. Quantitative HPLC determination of main flavonoid content of Rhododendron adamsii leaves and stems

    Komarova, N. I., Rogachev, A. D., Chernyak, E. I., Morozov, S. V., Fomenko, V. V. & Salakhutdinov, N. F., Jan 2009, In: Chemistry of Natural Compounds. 45, 1, p. 27-31 5 p.

    Research output: Contribution to journal › Article › peer-review

  192. 2006

  193. Comparative analysis of essential oil compositions from leaves and stems of Rhododendron adamsii, R. aureum, and R. dauricum

    Rogachev, A. D., Fomenko, V. V., Sal'nikova, O. I., Pokrovskii, L. M. & Salakhutdinov, N. F., Jul 2006, In: Chemistry of Natural Compounds. 42, 4, p. 426-430 5 p.

    Research output: Contribution to journal › Article › peer-review

ID: 3454033