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Fluorine-Containing n-6 and Angular and Linear n-6-n’ (n, n’ = 5, 6, 7) Diaza-Heterocyclic Scaffolds Assembled on Benzene Core in Unified Way. / Prima, Darya O.; Makarov, Arkady G.; Bagryanskaya, Irina Yu et al.

In: ChemistrySelect, Vol. 4, No. 8, 28.02.2019, p. 2383-2386.

Research output: Contribution to journal › Article › peer-review

Harvard

Prima, DO, Makarov, AG, Bagryanskaya, IY, Kolesnikov, AE, Zargarova, LV, Baev, DS, Eliseeva, TF, Politanskaya, LV, Makarov, AY, Slizhov, YG & Zibarev, AV 2019, 'Fluorine-Containing n-6 and Angular and Linear n-6-n’ (n, n’ = 5, 6, 7) Diaza-Heterocyclic Scaffolds Assembled on Benzene Core in Unified Way', ChemistrySelect, vol. 4, no. 8, pp. 2383-2386. https://doi.org/10.1002/slct.201803970

APA

Prima, D. O., Makarov, A. G., Bagryanskaya, I. Y., Kolesnikov, A. E., Zargarova, L. V., Baev, D. S., Eliseeva, T. F., Politanskaya, L. V., Makarov, A. Y., Slizhov, Y. G., & Zibarev, A. V. (2019). Fluorine-Containing n-6 and Angular and Linear n-6-n’ (n, n’ = 5, 6, 7) Diaza-Heterocyclic Scaffolds Assembled on Benzene Core in Unified Way. ChemistrySelect, 4(8), 2383-2386. https://doi.org/10.1002/slct.201803970

Vancouver

Prima DO, Makarov AG, Bagryanskaya IY, Kolesnikov AE, Zargarova LV, Baev DS et al. Fluorine-Containing n-6 and Angular and Linear n-6-n’ (n, n’ = 5, 6, 7) Diaza-Heterocyclic Scaffolds Assembled on Benzene Core in Unified Way. ChemistrySelect. 2019 Feb 28;4(8):2383-2386. doi: 10.1002/slct.201803970

Author

Prima, Darya O. ; Makarov, Arkady G. ; Bagryanskaya, Irina Yu et al. / Fluorine-Containing n-6 and Angular and Linear n-6-n’ (n, n’ = 5, 6, 7) Diaza-Heterocyclic Scaffolds Assembled on Benzene Core in Unified Way. In: ChemistrySelect. 2019 ; Vol. 4, No. 8. pp. 2383-2386.

BibTeX

@article{5ded7b3f86434a878bbce705a1586c20,
title = "Fluorine-Containing n-6 and Angular and Linear n-6-n{\textquoteright} (n, n{\textquoteright} = 5, 6, 7) Diaza-Heterocyclic Scaffolds Assembled on Benzene Core in Unified Way",
abstract = " The title compounds, including hybrids (n ≠ n{\textquoteright}), were assembled on benzene core in a unified way based on only one starting material C 6 F 5 NH 2 and a limited number of simple substitution and condensation reactions. The heterocyclic moieties were 1,3-diazoles, 1,2,3-triazoles, 1,2,5-thia(selena)diazoles, 1.4-diazines and 1,5-diazepines, as well as 1,3,2-dioxaboroles. Representatives of all new scaffolds were characterized by XRD. Compounds synthesized are of biomedical interest in the context of apoptotic anticancer activity, and the 1,2,5-thiadiazole/1,3,2-dioxaborole hybrid also in that of neutron or/and proton capture therapy of cancer. New 1,2,5-chalcogenadiazoles are protected forms of otherwise hardly accessible fluorine-containing di- and tetra-amines for further syntheses. ",
keywords = "benzo-fused heterocycles, boron heterocycles, fluoroaromatics, nitrogen heterocycles, structure elucidation, synthesis, ANIONS, PHARMACEUTICALS, COMPLEXES, MEDICINAL CHEMISTRY, METABOLISM, REDUCTION, CYCLIC ARYLENEAZACHALCOGENENES, QUINOXALINES, DERIVATIVES",
author = "Prima, {Darya O.} and Makarov, {Arkady G.} and Bagryanskaya, {Irina Yu} and Kolesnikov, {Andrey E.} and Zargarova, {Leila V.} and Baev, {Dmitry S.} and Eliseeva, {Tatiana F.} and Politanskaya, {Larisa V.} and Makarov, {Alexander Yu} and Slizhov, {Yuri G.} and Zibarev, {Andrey V.}",
year = "2019",
month = feb,
day = "28",
doi = "10.1002/slct.201803970",
language = "English",
volume = "4",
pages = "2383--2386",
journal = "ChemistrySelect",
issn = "2365-6549",
publisher = "Wiley-Blackwell",
number = "8",

}

RIS

TY - JOUR

T1 - Fluorine-Containing n-6 and Angular and Linear n-6-n’ (n, n’ = 5, 6, 7) Diaza-Heterocyclic Scaffolds Assembled on Benzene Core in Unified Way

AU - Prima, Darya O.

AU - Makarov, Arkady G.

AU - Bagryanskaya, Irina Yu

AU - Kolesnikov, Andrey E.

AU - Zargarova, Leila V.

AU - Baev, Dmitry S.

AU - Eliseeva, Tatiana F.

AU - Politanskaya, Larisa V.

AU - Makarov, Alexander Yu

AU - Slizhov, Yuri G.

AU - Zibarev, Andrey V.

PY - 2019/2/28

Y1 - 2019/2/28

N2 - The title compounds, including hybrids (n ≠ n’), were assembled on benzene core in a unified way based on only one starting material C 6 F 5 NH 2 and a limited number of simple substitution and condensation reactions. The heterocyclic moieties were 1,3-diazoles, 1,2,3-triazoles, 1,2,5-thia(selena)diazoles, 1.4-diazines and 1,5-diazepines, as well as 1,3,2-dioxaboroles. Representatives of all new scaffolds were characterized by XRD. Compounds synthesized are of biomedical interest in the context of apoptotic anticancer activity, and the 1,2,5-thiadiazole/1,3,2-dioxaborole hybrid also in that of neutron or/and proton capture therapy of cancer. New 1,2,5-chalcogenadiazoles are protected forms of otherwise hardly accessible fluorine-containing di- and tetra-amines for further syntheses.

AB - The title compounds, including hybrids (n ≠ n’), were assembled on benzene core in a unified way based on only one starting material C 6 F 5 NH 2 and a limited number of simple substitution and condensation reactions. The heterocyclic moieties were 1,3-diazoles, 1,2,3-triazoles, 1,2,5-thia(selena)diazoles, 1.4-diazines and 1,5-diazepines, as well as 1,3,2-dioxaboroles. Representatives of all new scaffolds were characterized by XRD. Compounds synthesized are of biomedical interest in the context of apoptotic anticancer activity, and the 1,2,5-thiadiazole/1,3,2-dioxaborole hybrid also in that of neutron or/and proton capture therapy of cancer. New 1,2,5-chalcogenadiazoles are protected forms of otherwise hardly accessible fluorine-containing di- and tetra-amines for further syntheses.

KW - benzo-fused heterocycles

KW - boron heterocycles

KW - fluoroaromatics

KW - nitrogen heterocycles

KW - structure elucidation

KW - synthesis

KW - ANIONS

KW - PHARMACEUTICALS

KW - COMPLEXES

KW - MEDICINAL CHEMISTRY

KW - METABOLISM

KW - REDUCTION

KW - CYCLIC ARYLENEAZACHALCOGENENES

KW - QUINOXALINES

KW - DERIVATIVES

UR - http://www.scopus.com/inward/record.url?scp=85062221121&partnerID=8YFLogxK

U2 - 10.1002/slct.201803970

DO - 10.1002/slct.201803970

M3 - Article

AN - SCOPUS:85062221121

VL - 4

SP - 2383

EP - 2386

JO - ChemistrySelect

JF - ChemistrySelect

SN - 2365-6549

IS - 8

ER -

ID: 18678310