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Synthesis and Antibacterial Activity of Caffeine Derivatives Containing Amino-Acid Fragments. / Reshetnikov, D. V.; Burova, L. G.; Rybalova, T. V. et al.

In: Chemistry of Natural Compounds, Vol. 58, No. 5, 09.2022, p. 908-915.

Research output: Contribution to journal › Article › peer-review

Harvard

Reshetnikov, DV, Burova, LG, Rybalova, TV, Bondareva, EA, Patrushev, SS, Evstropov, AN & Shults, EE 2022, 'Synthesis and Antibacterial Activity of Caffeine Derivatives Containing Amino-Acid Fragments', Chemistry of Natural Compounds, vol. 58, no. 5, pp. 908-915. https://doi.org/10.1007/s10600-022-03826-3

APA

Reshetnikov, D. V., Burova, L. G., Rybalova, T. V., Bondareva, E. A., Patrushev, S. S., Evstropov, A. N., & Shults, E. E. (2022). Synthesis and Antibacterial Activity of Caffeine Derivatives Containing Amino-Acid Fragments. Chemistry of Natural Compounds, 58(5), 908-915. https://doi.org/10.1007/s10600-022-03826-3

Vancouver

Reshetnikov DV, Burova LG, Rybalova TV, Bondareva EA, Patrushev SS, Evstropov AN et al. Synthesis and Antibacterial Activity of Caffeine Derivatives Containing Amino-Acid Fragments. Chemistry of Natural Compounds. 2022 Sept;58(5):908-915. doi: 10.1007/s10600-022-03826-3

Author

Reshetnikov, D. V. ; Burova, L. G. ; Rybalova, T. V. et al. / Synthesis and Antibacterial Activity of Caffeine Derivatives Containing Amino-Acid Fragments. In: Chemistry of Natural Compounds. 2022 ; Vol. 58, No. 5. pp. 908-915.

BibTeX

@article{bb3c76d3a825420d890b3b0242e1edca,
title = "Synthesis and Antibacterial Activity of Caffeine Derivatives Containing Amino-Acid Fragments",
abstract = "Cross-coupling of 8-bromocaffeine, 8-bromo-1-butyltheobromine, or 8-bromo-7-butyltheophylline with α-, β-, or ω-amino-acid methyl or t-butyl ester hydrochlorides in toluene in the presence of the catalytic system Pd(OAc)2·XantPhos and Cs2CO3 with microwave activation led to the formation of xanthine derivatives containing amino-acid fragments in the C-8 position. The antibacterial activity against Staphylococcus aureus and Bacillus cereus was studied.",
keywords = "amino acids, antibacterial activity, caffeine, catalytic amination, xanthines",
author = "Reshetnikov, {D. V.} and Burova, {L. G.} and Rybalova, {T. V.} and Bondareva, {E. A.} and Patrushev, {S. S.} and Evstropov, {A. N.} and Shults, {E. E.}",
note = "Funding Information: The work was financially supported by a Russian Science Foundation Grant (Project No. 18-13-00361). We thank the Khimiya Common Use Center, NIOCh, SB, RAS, for the spectral and analytical studies. Publisher Copyright: {\textcopyright} 2022, Springer Science+Business Media, LLC, part of Springer Nature.",
year = "2022",
month = sep,
doi = "10.1007/s10600-022-03826-3",
language = "English",
volume = "58",
pages = "908--915",
journal = "Chemistry of Natural Compounds",
issn = "0009-3130",
publisher = "Springer New York",
number = "5",

}

RIS

TY - JOUR

T1 - Synthesis and Antibacterial Activity of Caffeine Derivatives Containing Amino-Acid Fragments

AU - Reshetnikov, D. V.

AU - Burova, L. G.

AU - Rybalova, T. V.

AU - Bondareva, E. A.

AU - Patrushev, S. S.

AU - Evstropov, A. N.

AU - Shults, E. E.

N1 - Funding Information: The work was financially supported by a Russian Science Foundation Grant (Project No. 18-13-00361). We thank the Khimiya Common Use Center, NIOCh, SB, RAS, for the spectral and analytical studies. Publisher Copyright: © 2022, Springer Science+Business Media, LLC, part of Springer Nature.

PY - 2022/9

Y1 - 2022/9

N2 - Cross-coupling of 8-bromocaffeine, 8-bromo-1-butyltheobromine, or 8-bromo-7-butyltheophylline with α-, β-, or ω-amino-acid methyl or t-butyl ester hydrochlorides in toluene in the presence of the catalytic system Pd(OAc)2·XantPhos and Cs2CO3 with microwave activation led to the formation of xanthine derivatives containing amino-acid fragments in the C-8 position. The antibacterial activity against Staphylococcus aureus and Bacillus cereus was studied.

AB - Cross-coupling of 8-bromocaffeine, 8-bromo-1-butyltheobromine, or 8-bromo-7-butyltheophylline with α-, β-, or ω-amino-acid methyl or t-butyl ester hydrochlorides in toluene in the presence of the catalytic system Pd(OAc)2·XantPhos and Cs2CO3 with microwave activation led to the formation of xanthine derivatives containing amino-acid fragments in the C-8 position. The antibacterial activity against Staphylococcus aureus and Bacillus cereus was studied.

KW - amino acids

KW - antibacterial activity

KW - caffeine

KW - catalytic amination

KW - xanthines

UR - http://www.scopus.com/inward/record.url?scp=85138724857&partnerID=8YFLogxK

UR - https://www.mendeley.com/catalogue/7f6ce8da-a827-35a8-a1e7-99b996dff72c/

U2 - 10.1007/s10600-022-03826-3

DO - 10.1007/s10600-022-03826-3

M3 - Article

AN - SCOPUS:85138724857

VL - 58

SP - 908

EP - 915

JO - Chemistry of Natural Compounds

JF - Chemistry of Natural Compounds

SN - 0009-3130

IS - 5

ER -

ID: 38047591