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  1. 2019

  2. Novel inhibitors of DNA repair enzyme TDP1 combining monoterpenoid and adamantane fragments

    Mozhaitsev, E. S., Zakharenko, A. L., Suslov, E. V., Korchagina, D. V., Zakharova, O. D., Vasil’eva, I. A., Chepanova, A. A., Black, E., Patel, J., Chand, R., Reynisson, J., Leung, I. K. H., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jan 2019, In: Anti-Cancer Agents in Medicinal Chemistry. 19, 4, p. 463-472 10 p.

    Research output: Contribution to journal › Article › peer-review

  3. Novel tyrosyl-DNA phosphodiesterase 1 inhibitors enhance the therapeutic impact of topoteсan on in vivo tumor models

    Zakharenko, A. L., Luzina, O. A., Sokolov, D. N., Kaledin, V. I., Nikolin, V. P., Popova, N. A., Patel, J., Zakharova, O. D., Chepanova, A. A., Zafar, A., Reynisson, J., Leung, E., Leung, I. K. H., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jan 2019, In: European Journal of Medicinal Chemistry. 161, p. 581-593 13 p.

    Research output: Contribution to journal › Article › peer-review

  4. The development of tyrosyl-DNA phosphodyesterase 1 (TDP1) inhibitors based on the amines combining aromatic/heteroaromatic and monoterpenoid moieties

    Mozhaitsev, E., Suslov, E., Demidova, Y., Korchagina, D., Volcho, K., Zakharenko, A., Vasil’eva, I., Kupryushkin, M., Chepanova, A., Ayine-Tora, D. M., Reynisson, J., Salakhutdinov, N. & Lavrik, O., 1 Jan 2019, In: Letters in Drug Design and Discovery. 16, 5, p. 597-605 9 p.

    Research output: Contribution to journal › Article › peer-review

  5. Effects of acute and chronic treatment of STEP inhibitor, TC-2153, on the nervous system and behaviour of zebrafish (Danio rerio)

    Kulikov, A., Sinyakova, N., Kulikova, E., Evglevsky, N., Kolotygin, I., Volcho, K., Salakhutdinov, N., Kulikov, V., Romaschenko, A. & Moshkin, M., 2019, In: European Neuropsychopharmacology. 29, p. S198-S199 2 p.

    Research output: Contribution to journal › Meeting Abstract › peer-review

  6. 2018

  7. Molecular and Supramolecular Structure of 8-(Trifluoromethyl)Benzo[f][1,2,3,4,5] Pentathiepin-6-Amine – A Representative of Condensed Arene Pentathiepines

    Rybalova, T. V., Rogachev, A. D., Khomenko, T. M., Volcho, K. P. & Salakhutdinov, N. F., 1 Dec 2018, In: Journal of Structural Chemistry. 59, 7, p. 1753-1758 6 p.

    Research output: Contribution to journal › Article › peer-review

  8. Synthesis of d-(+)-camphor-based: N -acylhydrazones and their antiviral activity

    Kovaleva, K. S., Zubkov, F. I., Bormotov, N. I., Novikov, R. A., Dorovatovskii, P. V., Khrustalev, V. N., Gatilov, Y. V., Zarubaev, V. V., Yarovaya, O. I., Shishkina, L. N. & Salakhutdinov, N. F., 1 Dec 2018, In: MedChemComm. 9, 12, p. 2072-2082 11 p.

    Research output: Contribution to journal › Article › peer-review

  9. Untargeted search and identification of metabolites of antiviral agent camphecene in rat urine by liquid chromatography and mass spectrometry and studying their distribution in organs following peroral administration of the compound

    Rogachev, A. D., Yarovaya, O. I., Fatianova, A. V., Lavrinenko, V. A., Amosov, E. V., Zarubaev, V. V., Pokrovsky, A. G. & Salakhutdinov, N. F., 30 Nov 2018, In: Journal of Pharmaceutical and Biomedical Analysis. 161, p. 383-392 10 p.

    Research output: Contribution to journal › Article › peer-review

  10. Preparation of chiral isobenzofurans from 3-carene in the presence of modified clays

    Sidorenko, A. Y., Il'ina, I. V., Kravtsova, A. V., Aho, A., Ardashov, O. V., Li-Zhulanov, N. S., Volcho, K. P., Salakhutdinov, N. F., Murzin, D. Y. & Agabekov, V. E., 1 Nov 2018, In: Molecular Catalysis. 459, p. 38-45 8 p.

    Research output: Contribution to journal › Article › peer-review

  11. Selection of influenza virus resistant to the novel camphor-based antiviral camphecene results in loss of pathogenicity

    Zarubaev, V. V., Pushkina, E. A., Borisevich, S. S., Galochkina, A. V., Garshinina, A. V., Shtro, A. A., Egorova, A. A., Sokolova, A. S., Khursan, S. L., Yarovaya, O. I. & Salakhutdinov, N. F., 1 Nov 2018, In: Virology. 524, p. 69-77 9 p.

    Research output: Contribution to journal › Article › peer-review

  12. Highly selective reduction of nitroarenes by sc-isopropanol in the presence of zirconia in a flow reactor

    Anikeev, V. I., Sivcev, V. P., Valeev, K. R., Volcho, K. P., Sadykov, V. A. & Salakhutdinov, N. F., 1 Oct 2018, In: Journal of Supercritical Fluids. 140, p. 233-237 5 p.

    Research output: Contribution to journal › Article › peer-review

  13. Synthesis and antiviral activity of camphor-based 1,3-thiazolidin-4-one and thiazole derivatives as Orthopoxvirus-reproduction inhibitors

    Sokolova, A. S., Yarovaya, O. I., Bormotov, N. I., Shishkina, L. N. & Salakhutdinov, N. F., 1 Oct 2018, In: MedChemComm. 9, 10, p. 1746-1753 8 p.

    Research output: Contribution to journal › Article › peer-review

  14. A novel class of tyrosyl-DNA phosphodiesterase 1 inhibitors that contains the octahydro-2H-chromen-4-ol scaffold

    Li-Zhulanov, N. S., Zakharenko, A. L., Chepanova, A. A., Patel, J., Zafar, A., Volcho, K. P., Salakhutdinov, N. F., Reynisson, J., Leung, I. K. H. & Lavrik, O. I., 26 Sept 2018, In: Molecules. 23, 10, 14 p., 2468.

    Research output: Contribution to journal › Article › peer-review

  15. Discovery of a New Class of Inhibitors of Vaccinia Virus Based on (−)-Borneol from Abies sibirica and (+)-Camphor

    Sokolova, A. S., Yarovaya, O. I., Bormotov, N. I., Shishkina, L. N. & Salakhutdinov, N. F., 1 Sept 2018, In: Chemistry and Biodiversity. 15, 9, 9 p., e1800153.

    Research output: Contribution to journal › Article › peer-review

  16. Synthesis and evaluation of aryliden- and hetarylidenfuranone derivatives of usnic acid as highly potent Tdp1 inhibitors

    Zakharova, O., Luzina, O., Zakharenko, A., Sokolov, D., Filimonov, A., Dyrkheeva, N., Chepanova, A., Ilina, E., Ilyina, A., Klabenkova, K., Chelobanov, B., Stetsenko, D., Zafar, A., Eurtivong, C., Reynisson, J., Volcho, K., Salakhutdinov, N. & Lavrik, O., 15 Aug 2018, In: Bioorganic and Medicinal Chemistry. 26, 15, p. 4470-4480 11 p.

    Research output: Contribution to journal › Article › peer-review

  17. Synthesis and evaluation of camphor and cytisine-based cyanopyrrolidines as DPP-IV inhibitors for the treatment of type 2 diabetes mellitus

    Kuranov, S. O., Tsypysheva, I. P., Khvostov, M. V., Zainullina, L. F., Borisevich, S. S., Vakhitova, Y. V., Luzina, O. A. & Salakhutdinov, N. F., 15 Aug 2018, In: Bioorganic and Medicinal Chemistry. 26, 15, p. 4402-4409 8 p.

    Research output: Contribution to journal › Article › peer-review

  18. Preparation of octahydro-2H-chromen-4-ol with analgesic activity from isopulegol and thiophene-2-carbaldehyde in the presence of acid-modified clays

    Sidorenko, A. Y., Kravtsova, A. V., Wärnå, J., Aho, A., Heinmaa, I., Il'ina, I. V., Ardashov, O. V., Volcho, K. P., Salakhutdinov, N. F., Murzin, D. Y. & Agabekov, V. E., 1 Jul 2018, In: Molecular Catalysis. 453, p. 139-148 10 p.

    Research output: Contribution to journal › Article › peer-review

  19. Synthesis and Inhibitory Properties of Imines Containing Monoterpenoid and Adamantane Fragments Against DNA Repair Enzyme Tyrosyl-DNA Phosphodiesterase 1 (Tdp1)

    Zakharenko, A. L., Mozhaitsev, E. S., Suslov, E. V., Korchagina, D. V., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jul 2018, In: Chemistry of Natural Compounds. 54, 4, p. 672-676 5 p.

    Research output: Contribution to journal › Article › peer-review

  20. Highly potent activity of isopulegol-derived substituted octahydro-2H-chromen-4-ols against influenza A and B viruses

    Ilyina, I. V., Zarubaev, V. V., Lavrentieva, I. N., Shtro, A. A., Esaulkova, I. L., Korchagina, D. V., Borisevich, S. S., Volcho, K. P. & Salakhutdinov, N. F., 15 Jun 2018, In: Bioorganic and Medicinal Chemistry Letters. 28, 11, p. 2061-2067 7 p.

    Research output: Contribution to journal › Article › peer-review

  21. Usnic acid and its derivatives for pharmaceutical use: a patent review (2000–2017)

    Luzina, O. A. & Salakhutdinov, N. F., 3 Jun 2018, In: Expert Opinion on Therapeutic Patents. 28, 6, p. 477-491 15 p.

    Research output: Contribution to journal › Review article › peer-review

  22. 3-N-ЗАМЕЩЕННЫЕ БОРНИЛПРОПИОНАТЫ, ИСПОЛЬЗУЕМЫЕ В КАЧЕСТВЕ ИНГИБИТОРОВ ВИРУСА МАРБУРГ

    Яровая, О. И., Соколова, А. С., Кононова, А. А., Чересиз, С. В., Никитина, Р. А., Чепурнов, А. А., Зайковская, А. В., Пьянков, О. В., Покровский, А. Г., Максютов, Р. А. & Салахутдинов, Н. Ф., 3 Apr 2018, IPC No. A61K31/4453, A61K31/452, A61P31/12, C07D211/14, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2649406, Priority date 21 Sept 2017, Priority No. 2017133088

    Research output: Patent › Patent for invention

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