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Synthesis of 5-methyl-4-polyfluoroaryl-1,3-thiazol-2-amines. / Kalashnikov, Stepan B.; Vinogradov, Andrey S.; Yu. Bagryanskaya, Irina et al.

In: Mendeleev Communications, Vol. 34, No. 2, 01.03.2024, p. 277-278.

Research output: Contribution to journal › Article › peer-review

Harvard

Kalashnikov, SB, Vinogradov, AS, Yu. Bagryanskaya, I & Mezhenkova, TV 2024, 'Synthesis of 5-methyl-4-polyfluoroaryl-1,3-thiazol-2-amines', Mendeleev Communications, vol. 34, no. 2, pp. 277-278. https://doi.org/10.1016/j.mencom.2024.02.038

APA

Kalashnikov, S. B., Vinogradov, A. S., Yu. Bagryanskaya, I., & Mezhenkova, T. V. (2024). Synthesis of 5-methyl-4-polyfluoroaryl-1,3-thiazol-2-amines. Mendeleev Communications, 34(2), 277-278. https://doi.org/10.1016/j.mencom.2024.02.038

Vancouver

Kalashnikov SB, Vinogradov AS, Yu. Bagryanskaya I, Mezhenkova TV. Synthesis of 5-methyl-4-polyfluoroaryl-1,3-thiazol-2-amines. Mendeleev Communications. 2024 Mar 1;34(2):277-278. doi: 10.1016/j.mencom.2024.02.038

Author

Kalashnikov, Stepan B. ; Vinogradov, Andrey S. ; Yu. Bagryanskaya, Irina et al. / Synthesis of 5-methyl-4-polyfluoroaryl-1,3-thiazol-2-amines. In: Mendeleev Communications. 2024 ; Vol. 34, No. 2. pp. 277-278.

BibTeX

@article{0af72818ce2a404990ff573105270e15,
title = "Synthesis of 5-methyl-4-polyfluoroaryl-1,3-thiazol-2-amines",
abstract = "1-(Polyfluoroaryl)propan-1-ones were transformed into 5-methyl-4-polyfluoroaryl-1,3-thiazol-2-amines by a twostep reaction sequence involving formation of 2-bromo-1- (polyfluoroaryl)propan-1-ones under the acidic bromination conditions followed by heterocyclization with thiourea to finally afford new 5-methyl-4-polyfluoroaryl-1,3-thiazol-2- amines in high yields. 1,1'-(2,3,5,6-Tetrafluoro-1,4-phenylene)- dipropan-1-one was involved in the similar reaction to give a derivative containing two thiazole moieties.",
keywords = "X-ray diffraction analysis, bromination, organofluorine compounds, thiazoles, thiourea, α-bromo ketones",
author = "Kalashnikov, {Stepan B.} and Vinogradov, {Andrey S.} and {Yu. Bagryanskaya}, Irina and Mezhenkova, {Tatyana V.}",
note = "This work was supported by the Russian Science Foundation (grant no. 23-23-00547).",
year = "2024",
month = mar,
day = "1",
doi = "10.1016/j.mencom.2024.02.038",
language = "English",
volume = "34",
pages = "277--278",
journal = "Mendeleev Communications",
issn = "0959-9436",
publisher = "Elsevier",
number = "2",

}

RIS

TY - JOUR

T1 - Synthesis of 5-methyl-4-polyfluoroaryl-1,3-thiazol-2-amines

AU - Kalashnikov, Stepan B.

AU - Vinogradov, Andrey S.

AU - Yu. Bagryanskaya, Irina

AU - Mezhenkova, Tatyana V.

N1 - This work was supported by the Russian Science Foundation (grant no. 23-23-00547).

PY - 2024/3/1

Y1 - 2024/3/1

N2 - 1-(Polyfluoroaryl)propan-1-ones were transformed into 5-methyl-4-polyfluoroaryl-1,3-thiazol-2-amines by a twostep reaction sequence involving formation of 2-bromo-1- (polyfluoroaryl)propan-1-ones under the acidic bromination conditions followed by heterocyclization with thiourea to finally afford new 5-methyl-4-polyfluoroaryl-1,3-thiazol-2- amines in high yields. 1,1'-(2,3,5,6-Tetrafluoro-1,4-phenylene)- dipropan-1-one was involved in the similar reaction to give a derivative containing two thiazole moieties.

AB - 1-(Polyfluoroaryl)propan-1-ones were transformed into 5-methyl-4-polyfluoroaryl-1,3-thiazol-2-amines by a twostep reaction sequence involving formation of 2-bromo-1- (polyfluoroaryl)propan-1-ones under the acidic bromination conditions followed by heterocyclization with thiourea to finally afford new 5-methyl-4-polyfluoroaryl-1,3-thiazol-2- amines in high yields. 1,1'-(2,3,5,6-Tetrafluoro-1,4-phenylene)- dipropan-1-one was involved in the similar reaction to give a derivative containing two thiazole moieties.

KW - X-ray diffraction analysis

KW - bromination

KW - organofluorine compounds

KW - thiazoles

KW - thiourea

KW - α-bromo ketones

UR - https://www.scopus.com/record/display.uri?eid=2-s2.0-85189533262&origin=inward&txGid=9d22ca6eb29ade82bca4f598482bda47

UR - https://www.mendeley.com/catalogue/bf4b6522-cae3-39e2-846e-655f582df737/

U2 - 10.1016/j.mencom.2024.02.038

DO - 10.1016/j.mencom.2024.02.038

M3 - Article

VL - 34

SP - 277

EP - 278

JO - Mendeleev Communications

JF - Mendeleev Communications

SN - 0959-9436

IS - 2

ER -

ID: 61124480