1. 2021
  2. Design, synthesis, and molecular docking study of new tyrosyl-dna phosphodiesterase 1 (Tdp1) inhibitors combining resin acids and adamantane moieties

    Kovaleva, K., Yarovaya, O., Ponomarev, K., Cheresiz, S., Azimirad, A., Chernyshova, I., Zakharenko, A., Konev, V., Khlebnikova, T., Mozhaytsev, E., Suslov, E., Nilov, D., Švedas, V., Pokrovsky, A., Lavrik, O. & Salakhutdinov, N., 1 May 2021, In: Pharmaceuticals. 14, 5, 422.

    Research output: Contribution to journalArticlepeer-review

  3. Discovery of Novel Sultone Fused Berberine Derivatives as Promising Tdp1 Inhibitors

    Gladkova, E. D., Chepanova, A. A., Ilina, E. S., Zakharenko, A. L., Reynisson, J., Luzina, O. A., Volcho, K. P., Lavrik, O. I. & Salakhutdinov, N. F., 30 Mar 2021, In: Molecules (Basel, Switzerland). 26, 7, 1945.

    Research output: Contribution to journalArticlepeer-review

  4. Противоопухлевая активность комбинации топотекана и ингибитора тирозил-ДНК-фосфодиэстеразы 1 на модели асцитной карциномы Кребс-2 мыши

    Dyrkheeva, N. S., Zakharenko, A. L., Novoselova, E. S., Chepanova, A. A., Popova, N. A., Nikolin, V. P., Luzina, O. A., Salakhutdinov, N. F., Ryabchikova, E. I. & Lavrik, O. I., 1 Mar 2021, In: Molekuliarnaia biologiia. 55, 2, p. 312-317 6 p., 12.

    Research output: Contribution to journalArticlepeer-review

  5. Antitumor Activity of the Combination of Topotecan and Tyrosyl-DNA-Phosphodiesterase 1 Inhibitor on Model Krebs-2 Mouse Ascite Carcinoma

    Dyrkheeva, N. S., Zakharenko, A. L., Novoselova, E. S., Chepanova, A. A., Popova, N. A., Nikolin, V. P., Luzina, O. A., Salakhutdinov, N. F., Ryabchikova, E. I. & Lavrik, O. I., Mar 2021, In: Molecular Biology. 55, 2, p. 273-277 5 p.

    Research output: Contribution to journalArticlepeer-review

  6. Unexpected Ring Opening During the Imination of Camphor-Type Bicyclic Ketones

    Chernyshov, V. V., Yarovaya, O. I., Vatsadze, S. Z., Borisevich, S. S., Trukhan, S. N., Gatilov, Y. V., Peshkov, R. Y., Eltsov, I. V., Martyanov, O. N. & Salakhutdinov, N. F., 22 Jan 2021, In: European Journal of Organic Chemistry. 2021, 3, p. 452-463 12 p.

    Research output: Contribution to journalArticlepeer-review

  7. 2020
  8. Monoterpenoid-based inhibitors of filoviruses targeting the glycoprotein-mediated entry process

    Sokolova, A. S., Yarovaya, O. I., Zybkina, A. V., Mordvinova, E. D., Shcherbakova, N. S., Zaykovskaya, A. V., Baev, D. S., Tolstikova, T. G., Shcherbakov, D. N., Pyankov, O. V., Maksyutov, R. A. & Salakhutdinov, N. F., 1 Dec 2020, In: European Journal of Medicinal Chemistry. 207, 17 p., 112726.

    Research output: Contribution to journalArticlepeer-review

  9. The first berberine-based inhibitors of tyrosyl-dna phosphodiesterase 1 (Tdp1), an important dna repair enzyme

    Gladkova, E. D., Nechepurenko, I. V., Bredikhin, R. A., Chepanova, A. A., Zakharenko, A. L., Luzina, O. A., Ilina, E. S., Dyrkheeva, N. S., Mamontova, E. M., Anarbaev, R. O., Reynisson, J., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Oct 2020, In: International Journal of Molecular Sciences. 21, 19, p. 1-16 16 p., 7162.

    Research output: Contribution to journalArticlepeer-review

  10. New chemical agents based on adamantane-monoterpene conjugates against orthopoxvirus infections

    Suslov, E. V., Mozhaytsev, E. S., Korchagina, D. V., Bormotov, N. I., Yarovaya, O. I., Volcho, K. P., Serova, O. A., Agafonov, A. P., Maksyutov, R. A., Shishkina, L. N. & Salakhutdinov, N. F., Oct 2020, In: RSC Medicinal Chemistry. 11, 10, p. 1185-1195 11 p.

    Research output: Contribution to journalArticlepeer-review

  11. Menthylamine synthesis via gold-catalyzed hydrogenation of menthone oxime

    Demidova, Y. S., Mozhaitsev, E. S., Suslov, E. V., Nefedov, A. A., Saraev, A. A., Volcho, K. P., Salakhutdinov, N. F., Simakov, A., Simakova, I. L. & Murzin, D. Y., 5 Sept 2020, In: Applied Catalysis A: General. 605, 10 p., 117799.

    Research output: Contribution to journalArticlepeer-review

  12. Usnic Acid Conjugates with Monoterpenoids as Potent Tyrosyl-DNA Phosphodiesterase 1 Inhibitors

    Luzina, O., Filimonov, A., Zakharenko, A., Chepanova, A., Zakharova, O., Ilina, E., Dyrkheeva, N., Likhatskaya, G., Salakhutdinov, N. & Lavrik, O., 28 Aug 2020, In: Journal of Natural Products. 83, 8, p. 2320-2329 10 p.

    Research output: Contribution to journalArticlepeer-review

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