1. 2024
  2. 2-Aryl-1-hydroxyimidazoles possessing antiviral activity against a wide range of orthopoxviruses, including the variola virus

    Басанова, Е. И., Куликова, Е. А., Бормотов, Н. И., Серова, О. А., Шишкина, Л. Н., Овчинникова, А. С., Одношевский, Д. А., Пьянков, О. В., Агафонов, А. П., Яровая, О. И., Борисевич, С. С., Ильина, М. Г., Колыбалов, Д. С., Архипов, С. Г., Богданов, Н. Е., Павлова, М. А., Салахутдинов, Н. Ф., Перевалов, В. П. & Никитина, П. А., 5 Jul 2024, In: RSC Medicinal Chemistry. 15, 9, p. 3196-3211 16 p.

    Research output: Contribution to journalArticlepeer-review

  3. Производные имидазолидин-2,4-диона и имидазолидин-2,4,5-триона на основе смоляных кислот, проявляющие антиинвазивную активность в отношении клеток глиобластомы линий T98G и SNB19

    Чересиз, С. В., Ковалева, К. С., Яровая, О. И., Салахутдинов, Н. Ф. & Покровский, А. Г., 17 Jun 2024, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2821104, 8 Dec 2023, Priority date 8 Dec 2023, Priority No. 2023132332

    Research output: PatentPatent for invention

  4. Метаболомный скрининг методом ВЭЖХ-МС/МС в изучении биологических эффектов рентгеновского и терагерцового ЭМИ

    Басов, Н. В., Рогачев, А. Д., Бутикова, Е. А., Алешкова, М. А., Сотникова, М., Гайслер, Е. В., Яровая, О. И., Попик, В. М., Толстикова, Т. Г., Разумов, И. А., Покровский, А. Г. & Салахутдинов, Н. Ф., 2024, СИНХРОТРОННОЕ ИЗЛУЧЕНИЕ И ЛАЗЕРЫ НА СВОБОДНЫХ ЭЛЕКТРОНАХ (СИ И ЛСЭ - 2024): Книга тезисов. Новосибирск, p. 23-24

    Research output: Chapter in Book/Report/Conference proceedingConference contributionResearch

  5. 2023
  6. A Novel 3-meta-Pyridine-1,2,4-oxadiazole Derivative of Glycyrrhetinic Acid as a Safe and Promising Candidate for Overcoming P-Glycoprotein-Mediated Multidrug Resistance in Tumor Cells

    Moralev, A. D., Salomatina, O. V., Chernikov, I. V., Salakhutdinov, N. F., Zenkova, M. A. & Markov, A. V., 26 Dec 2023, In: ACS Omega. 8, 51, p. 48813-48824 12 p.

    Research output: Contribution to journalArticlepeer-review

  7. Pharmacokinetic study of Tdp1 inhibitor resulted in a significant increase in antitumor effect in the treatment of Lewis lung carcinoma in mice by its combination with topotecan

    Okhina, A. A., Kornienko, T. E., Rogachev, A. D., Luzina, O. A., Popova, N. A., Nikolin, V. P., Zakharenko, A. L., Dyrkheeva, N. S., Pokrovsky, A. G., Salakhutdinov, N. F. & Lavrik, O. I., 30 Nov 2023, In: Journal of Pharmaceutical and Biomedical Analysis. 236, 9 p., 115731.

    Research output: Contribution to journalArticlepeer-review

  8. Chiral N-(dialkyloctahydro-2H-chromen-4-yl)acetamides: synthesis and analgesic activity

    Li-Zhulanov, N. S., Kuznetsova, V. A., Gatilov, Y. V., Volcho, K. P., Khvostov, M. V., Tolstikova, T. G. & Salakhutdinov, N. F., Oct 2023, In: Russian Chemical Bulletin. 72, 10, p. 2430-2438 9 p.

    Research output: Contribution to journalArticlepeer-review

  9. Development of an LC-MS/MS-based method for quantification and pharmacokinetics study on SCID mice of a dehydroabietylamine-adamantylamine conjugate, a promising inhibitor of the DNA repair enzyme

    Okhina, A. A., Rogachev, A. D., Kovaleva, K. S., Yarovaya, O. I., Khotskina, A. S., Zavyalov, E. L., Vatsadze, S. Z., Pokrovsky, A. G. & Salakhutdinov, N. F., 20 Sept 2023, In: Journal of Pharmaceutical and Biomedical Analysis. 234, 115507.

    Research output: Contribution to journalArticlepeer-review

  10. Chiral N-(Octahydro-2H-chromen-4-yl)-2-(dialkylamino)acetamides: Synthesis and Analgesic Activity

    Li-Zhulanov, N. S., Nikolaichuk, K. M., Gatilov, Y. V., Volcho, K. P., Khvostov, M. V., Tolstikova, T. G. & Salakhutdinov, N. F., Sept 2023, In: Doklady Chemistry. 512, 1, p. 242-248 7 p.

    Research output: Contribution to journalArticlepeer-review

  11. Effect of Usnic Acid-Derived Tyrosyl-DNA Phosphodiesterase 1 Inhibitor Used as Monotherapy or in Combination with Olaparib on Transplanted Tumors In Vivo

    Kornienko, T. E., Zakharenko, A. L., Ilina, E. S., Chepanova, A. A., Zakharova, O. D., Dyrkheeva, N. S., Popova, N. A., Nikolin, V. P., Filimonov, A. S., Luzina, O. A., Salakhutdinov, N. F. & Lavrik, O. I., Apr 2023, In: Molecular Biology. 57, 2, p. 214-224 11 p.

    Research output: Contribution to journalArticlepeer-review

  12. Transcriptomic Analysis of CRISPR/Cas9-Mediated PARP1-Knockout Cells under the Influence of Topotecan and TDP1 Inhibitor

    Dyrkheeva, N. S., Malakhova, A. A., Zakharenko, A. L., Okorokova, L. S., Shtokalo, D. N., Pavlova, S. V., Medvedev, S. P., Zakian, S. M., Nushtaeva, A. A., Tupikin, A. E., Kabilov, M. R., Khodyreva, S. N., Luzina, O. A., Salakhutdinov, N. F. & Lavrik, O. I., 7 Mar 2023, In: International Journal of Molecular Sciences. 24, 6, 5148.

    Research output: Contribution to journalArticlepeer-review

  13. Synthesis of a Novel 9-O Berberine Derivative and Evaluation of Its Hypoglycemic Effect

    Gladkova, E. D., Valutsa, N., Borisov, S. A., Khvostov, M. V., Luzina, O. A., Tolstikova, T. G. & Salakhutdinov, N. F., Mar 2023, In: MolBank. 2023, 1, М1597.

    Research output: Contribution to journalArticlepeer-review

  14. Synthesis of N-heterocyclic amides based on (+)-camphoric acid and study of their antiviral activity and pharmacokinetics

    Yarovaya, O. I., Baranova, D. V., Sokolova, A. S., Nemolochnova, A. G., Sal'nikova, O. P., Fat'anova, A. V., Rogachev, A. D., Volobueva, A. S., Zarubaev, V. V., Pokrovsky, A. G. & Salakhutdinov, N. F., Mar 2023, In: Russian Chemical Bulletin. 72, 3, p. 807-818 12 p.

    Research output: Contribution to journalArticlepeer-review

  15. Novel TDP1 Inhibitors: Disubstituted Thiazolidine-2,4-Diones Containing Monoterpene Moieties

    Ivankin, D. I., Kornienko, T. E., Mikhailova, M. A., Dyrkheeva, N. S., Zakharenko, A. L., Achara, C., Reynisson, J., Golyshev, V. M., Luzina, O. A., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 14 Feb 2023, In: International Journal of Molecular Sciences. 24, 4, 3834.

    Research output: Contribution to journalArticlepeer-review

  16. 9-N-n-alkyl Berberine Derivatives: Hypoglycemic Activity Evaluation

    Khvostov, M. V., Gladkova, E. D., Borisov, S. A., Fedotova, M. S., Zhukova, N. A., Marenina, M. K., Meshkova, Y. V., Valutsa, N., Luzina, O. A., Tolstikova, T. G. & Salakhutdinov, N. F., 1 Jan 2023, In: Pharmaceutics. 15, 1, 44.

    Research output: Contribution to journalArticlepeer-review

  17. Structure-Based Design, Synthesis, and Biological Evaluation of the Cage-Amide Derived Orthopox Virus Replication Inhibitors

    Mozhaitsev, E. S., Suslov, E. V., Rastrepaeva, D. A., Yarovaya, O. I., Borisevich, S. S., Khamitov, E. M., Kolybalov, D. S., Arkhipov, S. G., Bormotov, N. I., Shishkina, L. N., Serova, O. A., Brunilin, R. V., Vernigora, A. A., Nawrozkij, M. B., Agafonov, A. P., Maksyutov, R. A., Volcho, K. P. & Salakhutdinov, N. F., 1 Jan 2023, In: Viruses. 15, 1, 29.

    Research output: Contribution to journalArticlepeer-review

  18. Synthesis of conjugates of (aR,7S)-colchicine with monoterpenoids and investigation of their biological activity

    Shchegravina, E. S., Usova, S. D., Baev, D. S., Mozhaitsev, E. S., Shcherbakov, D. N., Belenkaya, S. V., Volosnikova, E. A., Chirkova, V. Y., Sharlaeva, E. A., Svirshchevskaya, E. V., Fonareva, I. P., Sitdikova, A. R., Salakhutdinov, N. F., Yarovaya, O. I. & Fedorov, A. Y., 1 Jan 2023, In: Russian Chemical Bulletin. 72, 1, p. 248-262 15 p.

    Research output: Contribution to journalArticlepeer-review

  19. Synthesis of non-symmetric N-benzylbispidinol amides and study of their inhibitory activity against the main protease of the SARS-CoV-2 virus

    Dalinger, A. I., Baev, D. S., Yarovaya, O. I., Chirkova, V. Y., Sharlaeva, E. A., Belenkaya, S. V., Shcherbakov, D. N., Salakhutdinov, N. F. & Vatsadze, S. Z., 1 Jan 2023, In: Russian Chemical Bulletin. 72, 1, p. 239-247 9 p.

    Research output: Contribution to journalArticlepeer-review

Previous 1 2 3 4 5 6 7 8 ...10 Next

ID: 3454033