1. 2019
  2. Novel inhibitors of DNA repair enzyme TDP1 combining monoterpenoid and adamantane fragments

    Mozhaitsev, E. S., Zakharenko, A. L., Suslov, E. V., Korchagina, D. V., Zakharova, O. D., Vasil’eva, I. A., Chepanova, A. A., Black, E., Patel, J., Chand, R., Reynisson, J., Leung, I. K. H., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jan 2019, In: Anti-Cancer Agents in Medicinal Chemistry. 19, 4, p. 463-472 10 p.

    Research output: Contribution to journalArticlepeer-review

  3. Novel tyrosyl-DNA phosphodiesterase 1 inhibitors enhance the therapeutic impact of topoteсan on in vivo tumor models

    Zakharenko, A. L., Luzina, O. A., Sokolov, D. N., Kaledin, V. I., Nikolin, V. P., Popova, N. A., Patel, J., Zakharova, O. D., Chepanova, A. A., Zafar, A., Reynisson, J., Leung, E., Leung, I. K. H., Volcho, K. P., Salakhutdinov, N. F. & Lavrik, O. I., 1 Jan 2019, In: European Journal of Medicinal Chemistry. 161, p. 581-593 13 p.

    Research output: Contribution to journalArticlepeer-review

  4. The development of tyrosyl-DNA phosphodyesterase 1 (TDP1) inhibitors based on the amines combining aromatic/heteroaromatic and monoterpenoid moieties

    Mozhaitsev, E., Suslov, E., Demidova, Y., Korchagina, D., Volcho, K., Zakharenko, A., Vasil’eva, I., Kupryushkin, M., Chepanova, A., Ayine-Tora, D. M., Reynisson, J., Salakhutdinov, N. & Lavrik, O., 1 Jan 2019, In: Letters in Drug Design and Discovery. 16, 5, p. 597-605 9 p.

    Research output: Contribution to journalArticlepeer-review

  5. Increasing bioavailability of very poorly water-soluble compounds. A case study of an anti-tumor drug, soloxolon methyl

    Ogienko, A. G., Markov, A. V., Sen'kova, A. V., Logashenko, E. B., Salomatina, O. V., Myz, S. A., Ogienko, A. A., Nefedov, A. A., Losev, E. A., Drebushchak, T. N., Salakhutdinov, N. F., Boldyrev, V. V., Vlasov, V. V., Zenkova, M. A. & Boldyreva, E. V., 1 Feb 2019, In: Journal of Drug Delivery Science and Technology. 49, p. 35-42 8 p.

    Research output: Contribution to journalArticlepeer-review

  6. Synthesis of diazaadamantanes from 1,5-dimethylbispidinone and some natural ketones

    Suslov, E. V., Ponomarev, K. Y., Korchagina, D. V., Volcho, K. P. & Salakhutdinov, N. F., 1 Mar 2019, In: Russian Chemical Bulletin. 68, 3, p. 601-605 5 p.

    Research output: Contribution to journalArticlepeer-review

  7. Antimetastatic Activity of Combined Topotecan and Tyrosyl-DNA Phosphodiesterase-1 Inhibitor on Modeled Lewis Lung Carcinoma

    Koldysheva, E. V., Men’shchikova, A. P., Lushnikova, E. L., Popova, N. A., Kaledin, V. I., Nikolin, V. P., Zakharenko, A. L., Luzina, O. A., Salakhutdinov, N. F. & Lavrik, O. I., 15 Mar 2019, In: Bulletin of Experimental Biology and Medicine. 166, 5, p. 661-666 6 p.

    Research output: Contribution to journalArticlepeer-review

  8. Effect of chiral polyhydrochromenes on cannabinoid system

    Li-Zhulanov, N. S., Il’ina, I. V., Chicca, A., Schenker, P., Patrusheva, O. S., Nazimova, E. V., Korchagina, D. V., Krasavin, M., Volcho, K. P. & Salakhutdinov, N. F., Apr 2019, In: Medicinal Chemistry Research. 28, 4, p. 450-464 15 p.

    Research output: Contribution to journalArticlepeer-review

  9. Synthesis and analgesic activity of octahydro-2H-chromenols, derivatives of aliphatic ketones

    Il’ina, I. V., Korchagina, D. V., Morozova, E. A., Tolstikova, T. G., Volcho, K. P. & Salakhutdinov, N. F., 1 May 2019, In: Russian Chemical Bulletin. 68, 5, p. 1061-1066 6 p.

    Research output: Contribution to journalArticlepeer-review

  10. Synthesis, hypolipidemic and antifungal activity of tetrahydroberberrubine sulfonates

    Nechepurenko, I. V., Shirokova, E. D., Khvostov, M. V., Frolova, T. S., Sinitsyna, O. I., Maksimov, A. M., Bredikhin, R. A., Komarova, N. I., Fadeev, D. S., Luzina, O. A., Tolstikova, T. G. & Salakhutdinova, N. F., 1 May 2019, In: Russian Chemical Bulletin. 68, 5, p. 1052-1060 9 p.

    Research output: Contribution to journalArticlepeer-review

  11. Synthesis of (1S)-(+)-camphor-10-sulfonic acid derivatives and investigations in vitro and in silico of their antiviral activity as the inhibitors of fi lovirus infections

    Sokolova, A. S., Baranova, D. V., Yarovaya, O. I., Baev, D. S., Polezhaeva, O. A., Zybkina, A. V., Shcherbakov, D. N., Tolstikova, T. G. & Salakhutdinov, N. F., 1 May 2019, In: Russian Chemical Bulletin. 68, 5, p. 1041-1046 6 p.

    Research output: Contribution to journalArticlepeer-review

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