1. 2026
  2. Bicyclic monoterpenoid-based orthopoxvirus inhibitors: Design, synthesis, and biological assessment of a novel amide series

    Tishchenko, S. A., Sokolova, A. S., Samsonova, V. V., Pushkareva, J. G., Bormotov, N. I., Moskalev, I. A., Solomina, D. E., Rogachev, A. D., Fatyanova, A. V., Borisevich, S. S., Yarovaya, O. I., Serova, O. A., Ovchinnikova, A. S., Sergeev, A. A., Shishkina, L. N., Sergeev, A. A., Agafonov, A. P. & Salakhutdinov, N. F., 9 Apr 2026, In: RSC Medicinal Chemistry. 17, 5, p. 2605-2629 25 p.

    Research output: Contribution to journal › Article › peer-review

  3. 2025
  4. Expanding the antiviral arsenal: N-arylated 1,2,4-oxadiazol-5(4H)-ones show high activity against orthopoxviruses

    Semenov, A. V., Baykov, S. V., Soldatova, N. S., Geyl, K. K., Shetnev, A. A., Boyarskiy, V. P., Yusubov, M. S., Bormotov, N. I., Serova, O. A., Shishkina, L. N., Ovchinnikova, A. S., Odnoshevsky, D. A., Pyankov, O. V., Borisevich, S. S., Gorohov, Y. V., Nikitin, V. N., Shcherbakov, D. N., Yarovaya, O. I., Salakhutdinov, N. F. & Postnikov, P. S., 15 Dec 2025, In: European Journal of Medicinal Chemistry. 300, p. 118124 16 p., 118124.

    Research output: Contribution to journal › Article › peer-review

  5. Biostability, in vivo antiviral activity against respiratory syncytial virus, and pharmacokinetic profiles of (−)-borneol esters

    Sokolova, A. S., Okhina, A. A., Shtro, A. A., Klabukov, A. M., Galochkina, A. V., Nikolaeva, Y. V., Petukhova, G. D., Yarovaya, O. I., Rogachev, A. D., Baev, D. S., Fatyanova, A. V., Tolstikova, T. G. & Salakhutdinov, N. F., 5 Jun 2025, In: European Journal of Pharmacology. 996, 177567.

    Research output: Contribution to journal › Article › peer-review

  6. Synthesis and a Kinetic Study of the Reactivity of 1-Amino-7,7-dimethylbicyclo[2.2.1]heptan-2-one in Alkylation Reactions with Structurally Similar Amines

    Tishchenko, S., Sokolova, A. S., Arbuzova, M. A., Selyutina, O. Y., Tsypyshev, D. O., Yarovaya, O. I., Arkhipov, S. G. & Salakhutdinov, N. F., 23 May 2025, In: ChemistrySelect. 10, 20, e05689.

    Research output: Contribution to journal › Article › peer-review

  7. Synthesis of Secondary Amines of Bornylamine and Isobornylamine Containing a Saturated N-Heterocycle and Study of Their Antiviral Activity against Respiratory Syncytial Virus

    Tishchenko, S. A., Sokolova, A. S., Yarovaya, O. I., Krasnov, V. I., Shtro, A. A., Galochkina, A. V., Klabukov, A. M., Razgulyaeva, D. N. & Salakhutdinov, N. F., 27 Feb 2025, In: Russian Journal of General Chemistry. 95, 1, p. 79-87 9 p.

    Research output: Contribution to journal › Article › peer-review

  8. New thiosemicarbazones possessing activity against SARS-CoV-2 and H1N1 influenza viruses

    Zhupikova, O. A., Yarovaya, O. I., Marenina, M. K., Meshkova, Y. V., Belenkaya, S. V., Shcherbakov, D. N., Zaykovskaya, A. V., Pyankov, O. V., Zarubaev, V. V., Mikhalsky, M. G., Fedorov, A. Y., Arkhipov, S. G., Potkin, V. I., Kolesnik, I. A., Ivanov, A. V., Salakhutdinov, N. F. & Khvostov, M. V., 2025, In: Mendeleev Communications. 35, 2, p. 145-147 3 p.

    Research output: Contribution to journal › Article › peer-review

  9. Радиозащитные свойства препарата «Димефосфон» на модели лучевого поражения in vivo

    Kiseleva, D. A., Melchenko, M. A., Yarovaya, O. I., Basov, N. V., Rogachev, A. D., Pokrovsky, A. G., Salakhutdinov, N. F. & Tolstikova, T. G., 2025, In: Acta Naturae. 17, 4, p. 93-102 10 p., 8.

    Research output: Contribution to journal › Article › peer-review

  10. 2024
  11. (+)-fenchol and (−)-isopinocampheol derivatives targeting the entry process of filoviruses

    Sokolova, A. S., Baev, D. S., Mordvinova, E. D., Yarovaya, O. I., Volkova, N. V., Shcherbakov, D. N., Okhina, A. A., Rogachev, A. D., Shnaider, T. A., Chvileva, A. S., Nikitina, T. V., Tolstikova, T. G. & Salakhutdinov, N. F., 5 Sept 2024, In: European Journal of Medicinal Chemistry. 275, 16 p., 116596.

    Research output: Contribution to journal › Article › peer-review

  12. 2-Aryl-1-hydroxyimidazoles possessing antiviral activity against a wide range of orthopoxviruses, including the variola virus

    Басанова, Е. И., Куликова, Е. А., Бормотов, Н. И., Серова, О. А., Шишкина, Л. Н., Овчинникова, А. С., Одношевский, Д. А., Пьянков, О. В., Агафонов, А. П., Яровая, О. И., Борисевич, С. С., Ильина, М. Г., Колыбалов, Д. С., Архипов, С. Г., Богданов, Н. Е., Павлова, М. А., Салахутдинов, Н. Ф., Перевалов, В. П. & Никитина, П. А., 5 Jul 2024, In: RSC Medicinal Chemistry. 15, 9, p. 3196-3211 16 p.

    Research output: Contribution to journal › Article › peer-review

  13. Производные имидазолидин-2,4-диона и имидазолидин-2,4,5-триона на основе смоляных кислот, проявляющие антиинвазивную активность в отношении клеток глиобластомы линий T98G и SNB19

    Чересиз, С. В., Ковалева, К. С., Яровая, О. И., Салахутдинов, Н. Ф. & Покровский, А. Г., 17 Jun 2024, Роспатент - Федеральная служба по интеллектуальной собственности, Patent No. 2821104, 8 Dec 2023, Priority date 8 Dec 2023, Priority No. 2023132332

    Research output: Patent › Patent for invention

  14. Метаболомный скрининг методом ВЭЖХ-МС/МС в изучении биологических эффектов рентгеновского и терагерцового ЭМИ

    Басов, Н. В., Рогачев, А. Д., Бутикова, Е. А., Алешкова, М. А., Сотникова, М., Гайслер, Е. В., Яровая, О. И., Попик, В. М., Толстикова, Т. Г., Разумов, И. А., Покровский, А. Г. & Салахутдинов, Н. Ф., 2024, СИНХРОТРОННОЕ ИЗЛУЧЕНИЕ И ЛАЗЕРЫ НА СВОБОДНЫХ ЭЛЕКТРОНАХ (СИ И ЛСЭ - 2024): Книга тезисов. Новосибирск, p. 23-24

    Research output: Chapter in Book/Report/Conference proceeding › Conference contribution › Research

  15. 2023
  16. Development of an LC-MS/MS-based method for quantification and pharmacokinetics study on SCID mice of a dehydroabietylamine-adamantylamine conjugate, a promising inhibitor of the DNA repair enzyme

    Okhina, A. A., Rogachev, A. D., Kovaleva, K. S., Yarovaya, O. I., Khotskina, A. S., Zavyalov, E. L., Vatsadze, S. Z., Pokrovsky, A. G. & Salakhutdinov, N. F., 20 Sept 2023, In: Journal of Pharmaceutical and Biomedical Analysis. 234, 115507.

    Research output: Contribution to journal › Article › peer-review

  17. Synthesis of N-heterocyclic amides based on (+)-camphoric acid and study of their antiviral activity and pharmacokinetics

    Yarovaya, O. I., Baranova, D. V., Sokolova, A. S., Nemolochnova, A. G., Sal'nikova, O. P., Fat'anova, A. V., Rogachev, A. D., Volobueva, A. S., Zarubaev, V. V., Pokrovsky, A. G. & Salakhutdinov, N. F., Mar 2023, In: Russian Chemical Bulletin. 72, 3, p. 807-818 12 p.

    Research output: Contribution to journal › Article › peer-review

  18. Structure-Based Design, Synthesis, and Biological Evaluation of the Cage-Amide Derived Orthopox Virus Replication Inhibitors

    Mozhaitsev, E. S., Suslov, E. V., Rastrepaeva, D. A., Yarovaya, O. I., Borisevich, S. S., Khamitov, E. M., Kolybalov, D. S., Arkhipov, S. G., Bormotov, N. I., Shishkina, L. N., Serova, O. A., Brunilin, R. V., Vernigora, A. A., Nawrozkij, M. B., Agafonov, A. P., Maksyutov, R. A., Volcho, K. P. & Salakhutdinov, N. F., 1 Jan 2023, In: Viruses. 15, 1, 29.

    Research output: Contribution to journal › Article › peer-review

  19. Synthesis of conjugates of (aR,7S)-colchicine with monoterpenoids and investigation of their biological activity

    Shchegravina, E. S., Usova, S. D., Baev, D. S., Mozhaitsev, E. S., Shcherbakov, D. N., Belenkaya, S. V., Volosnikova, E. A., Chirkova, V. Y., Sharlaeva, E. A., Svirshchevskaya, E. V., Fonareva, I. P., Sitdikova, A. R., Salakhutdinov, N. F., Yarovaya, O. I. & Fedorov, A. Y., 1 Jan 2023, In: Russian Chemical Bulletin. 72, 1, p. 248-262 15 p.

    Research output: Contribution to journal › Article › peer-review

  20. Synthesis of non-symmetric N-benzylbispidinol amides and study of their inhibitory activity against the main protease of the SARS-CoV-2 virus

    Dalinger, A. I., Baev, D. S., Yarovaya, O. I., Chirkova, V. Y., Sharlaeva, E. A., Belenkaya, S. V., Shcherbakov, D. N., Salakhutdinov, N. F. & Vatsadze, S. Z., 1 Jan 2023, In: Russian Chemical Bulletin. 72, 1, p. 239-247 9 p.

    Research output: Contribution to journal › Article › peer-review

  21. Corrigendum: The main protease 3CLpro of the SARS-CoV-2 virus: how to turn an enemy into a helper

    Belenkaya, S. V., Merkuleva, I. A., Yarovaya, O. I., Chirkova, V. Y., Sharlaeva, E. A., Shanshin, D. V., Volosnikova, E. A., Vatsadze, S. Z., Khvostov, M. V., Salakhutdinov, N. F. & Shcherbakov, D., 2023, In: Frontiers in Bioengineering and Biotechnology. 11, 1294266.

    Research output: Contribution to journal › Article › peer-review

  22. The main protease 3CLpro of the SARS-CoV-2 virus: how to turn an enemy into a helper

    Belenkaya, S. V., Merkuleva, I. A., Yarovaya, O. I., Chirkova, V. Y., Sharlaeva, E. A., Shanshin, D. V., Volosnikova, E. A., Vatsadze, S. Z., Khvostov, M. V., Salakhutdinov, N. F. & Shcherbakov, D. N., 2023, In: Frontiers in Bioengineering and Biotechnology. 11, 1187761.

    Research output: Contribution to journal › Article › peer-review

Previous 1 2 3 4 Next

ID: 3449511